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Ibrutinib targets mutant-EGFR kinase with a distinct binding conformation 期刊论文
ONCOTARGET, 2016, 卷号: 7, 期号: 43, 页码: 69760-69769
作者:  Wang, Aoli;  Yan, Xiao-E;  Wu, Hong;  Wang, Wenchao;  Hu, Chen;  Chen, Cheng;  Zhao, Zheng;  Zhao, Peng;  Li, Xixiang;  Wang, Li;  Wang, Beilei;  Ye, Zi;  Wang, Jinhua;  Wang, Chu;  Zhang, Wei;  Gray, Nathanael S.;  Weisberg, Ellen L.;  Chen, Liang;  Liu, Jing;  Yun, Cai-Hong;  Liu, Qingsong
浏览  |  Adobe PDF(2026Kb)  |  收藏  |  浏览/下载:124/63  |  提交时间:2017/11/21
Ibrutinib  Egfr Kinase  Dfg-in/c-helix-out  Inactive Conformation  Nsclc  
Discovery and characterization of a novel potent type II native and mutant BCR-ABL inhibitor (CHMFL-074) for Chronic Myeloid Leukemia (CML) 期刊论文
ONCOTARGET, 2016, 卷号: 7, 期号: 29, 页码: 45562-45574
作者:  Liu, Feiyang;  Wang, Beilei;  Wang, Qiang;  Qi, Ziping;  Chen, Cheng;  Kong, Lu-Lu;  Chen, Ji-Yun;  Liu, Xiaochuan;  Wang, Aoli;  Hu, Chen;  Wang, Wenchao;  Wang, Huiping;  Wu, Fan;  Ruan, Yanjie;  Qi, Shuang;  Liu, Juan;  Zou, Fengming;  Hu, Zhenquan;  Wang, Wei;  Wang, Li;  Zhang, Shanchun;  Yun, Cai-Hong;  Zhai, Zhimin;  Liu, Jing;  Liu, Qingsong
浏览  |  Adobe PDF(8054Kb)  |  收藏  |  浏览/下载:254/200  |  提交时间:2017/11/21
Bcr-abl  Pdgfr  Chronic Myeloid Leukemia  Kinase Inhibitor  
Moderate and strong static magnetic fields directly affect EGFR kinase domain orientation to inhibit cancer cell proliferation 期刊论文
ONCOTARGET, 2016, 卷号: 7, 期号: 27, 页码: 41527-41539
作者:  Zhang, Lei;  Wang, Jihao;  Wang, HongLei;  Wang, Wenchao;  Li, Zhiyuan;  Liu, Juanjuan;  Yang, Xingxing;  Ji, Xinmiao;  Luo, Yan;  Hu, Chen;  Hou, Yubin;  He, Qianqian;  Fang, Jun;  Wang, Junfeng;  Liu, Qingsong;  Li, Guohui;  Lu, Qingyou;  Zhang, Xin
浏览  |  Adobe PDF(11191Kb)  |  收藏  |  浏览/下载:103/43  |  提交时间:2017/11/21
Egfr  Magnetic Field  Stm  Cancer