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Injectable magnetic montmorillonite colloidal gel for the postoperative treatment of hepatocellular carcinoma 期刊论文
JOURNAL OF NANOBIOTECHNOLOGY, 2022, 卷号: 20
作者:  Chen, Sheng;  Song, Yonghong;  Yan, Xu;  Dong, Liang;  Xu, Yunjun;  Xuan, Shouhu;  Shu, Quan;  Cao, Baoqiang;  Hu, Jinlong;  Xing, Hanye;  Wu, Wenshu;  Zha, Zhengbao;  Lu, Yang
收藏  |  浏览/下载:38/0  |  提交时间:2022/12/23
Colloidal gel  Magnetic hyperthermia  Hepatocellular carcinoma  Postoperative therapy  Hemostasis  
CHMFL-26 is a highly potent irreversible HER2 inhibitor for use in the treatment of HER2-positive and HER2-mutant cancers 期刊论文
ACTA PHARMACOLOGICA SINICA, 2022
作者:  Cao, Jiang-yan;  Qi, Shuang;  Wu, Hong;  Wang, Ao-li;  Liu, Qing-wang;  Li, Xi-xiang;  Wang, Bei-lei;  Ge, Juan;  Zou, Feng-ming;  Chen, Cheng;  Wang, Jun-jie;  Hu, Chen;  Liu, Jing;  Wang, Wen-chao;  Liu, Qing-song
收藏  |  浏览/下载:104/0  |  提交时间:2022/03/28
HER2  breast cancers  gastric cancers  irreversible inhibitor  drug resistance  
An overview of kinase downregulators and recent advances in discovery approaches 期刊论文
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2021, 卷号: 6
作者:  Wang, Beilei;  Wu, Hong;  Hu, Chen;  Wang, Haizhen;  Liu, Jing;  Wang, Wenchao;  Liu, Qingsong
收藏  |  浏览/下载:76/0  |  提交时间:2022/01/25
CD71-Specific Aptamer Conjugated with Monomethyl Auristatin E for the Treatment of Uveal Melanoma 期刊论文
ACS APPLIED MATERIALS & INTERFACES, 2021
作者:  Zhang, Hui;  Jin, Cheng;  Zhang, Lin;  Peng, Bo;  Zhang, Yibin;  Liu, Yan;  Li, Ling;  Ye, Mao;  Xiong, Wei;  Tan, Weihong
收藏  |  浏览/下载:55/0  |  提交时间:2022/02/14
uveal melanoma  CD71  aptamer-drug conjugate  targeted drug delivery  tumor-targeted therapy  
Discovery of a highly potent and selective Bruton's tyrosine kinase inhibitor avoiding impairment of ADCC effects for B-cell non-Hodgkin lymphoma 期刊论文
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2020, 卷号: 5
作者:  Liu, Juan;  Liang, Qianmao;  Wang, Aoli;  Zou, Fengming;  Qi, Ziping;  Yu, Kailin;  Liu, Qingwang;  Chen, Cheng;  Liu, Jing;  Liu, Qingsong
收藏  |  浏览/下载:51/0  |  提交时间:2020/11/30
Design and test of superconducting magnet for 200 MeV proton cyclotron 期刊论文
CRYOGENICS, 2019, 卷号: 97, 期号: 无, 页码: 122-125
作者:  Du, S.;  Zou, C.;  Ding, K.;  Liu, X.;  Chen, Y.;  Song, Y.
浏览  |  Adobe PDF(959Kb)  |  收藏  |  浏览/下载:70/36  |  提交时间:2020/05/21
Proton cyclotron  Superconducting coil  Quench protection system  Energizing  
The Role of Endoplasmic Reticulum in Introducing Nano-toxicology and The Mechanism Involved 期刊论文
PROGRESS IN BIOCHEMISTRY AND BIOPHYSICS, 2019, 卷号: 46, 期号: 1, 页码: 20-31
作者:  Wang Juan;  Xu Wen-Juan;  Wang Xin-Wen;  Wang Jing-Jing;  Wang Mei-Mei;  Xu An
浏览  |  Adobe PDF(10635Kb)  |  收藏  |  浏览/下载:120/42  |  提交时间:2020/03/31
endoplasmic reticulum  nanomaterials  apoptosis  inflammation  autophagy  toxicity  
Repurposing cabozantinib to GISTs: Overcoming multiple imatinib-resistant cKIT mutations including gatekeeper and activation loop mutants in GISTs preclinical models 期刊论文
CANCER LETTERS, 2019, 页码: 105-114
作者:  Lu, Tingting;  Chen, Cheng;  Wang, Aoli;  Jiang, Zongru;  Qi, Ziping;  Hu, Zhenquan;  Hu, Chen;  Liu, Feiyang;  Wang, Wenliang;  Wu, Hong;  Wang, Beilei;  Wang, Li;  Qi, Shuang;  Wu, Jiaxin;  Wang, Wenchao;  Tang, Jun;  Yan, Hezhong;  Bai, Mingfeng;  Liu, Qingsong;  Liu, Jing
收藏  |  浏览/下载:26/0  |  提交时间:2020/07/14
cKIT T670I mutant  Activation loop mutants  Drug resistance  
Discovery of 4-(((4-(5-chloro-2-(((1s,4s)-4-((2-methoxyethyl)amino) cyclohexyl)amino)pyridin-4-yl)thiazol-2-yl)amino)methyl) tetrahydro-2H-pyran-4-carbonitrile (JSH-150) as a novel highly selective and potent CDK9 kinase inhibitor 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 158, 页码: 896-916
作者:  Wang, Beilei;  Wu, Jiaxin;  Wu, Yun;  Chen, Cheng;  Zou, Fengming;  Wang, Aoli;  Wu, Hong;  Hu, Zhenquan;  Jiang, Zongru;  Liu, Qingwang;  Wang, Wei;  Zhang, Yicong;  Liu, Feiyang;  Zhao, Ming;  Hu, Jie;  Huang, Tao;  Ge, Juan;  Wang, Li;  Ren, Tao;  Wang, Yuxin;  Liu, Jing;  Liu, Qingsong
收藏  |  浏览/下载:28/0  |  提交时间:2019/12/25
CDK9  Kinase inhibitor  Structure-activity relationship  Leukemia