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中国科学院合肥物质科学研究院机构知识库
Knowledge Management System of Hefei Institute of Physical Science,CAS
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CHMFL-26 is a highly potent irreversible HER2 inhibitor for use in the treatment of HER2-positive and HER2-mutant cancers
期刊论文
ACTA PHARMACOLOGICA SINICA, 2022
作者:
Cao, Jiang-yan
;
Qi, Shuang
;
Wu, Hong
;
Wang, Ao-li
;
Liu, Qing-wang
;
Li, Xi-xiang
;
Wang, Bei-lei
;
Ge, Juan
;
Zou, Feng-ming
;
Chen, Cheng
;
Wang, Jun-jie
;
Hu, Chen
;
Liu, Jing
;
Wang, Wen-chao
;
Liu, Qing-song
收藏
  |  
浏览/下载:104/0
  |  
提交时间:2022/03/28
HER2
breast cancers
gastric cancers
irreversible inhibitor
drug resistance
An overview of kinase downregulators and recent advances in discovery approaches
期刊论文
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2021, 卷号: 6
作者:
Wang, Beilei
;
Wu, Hong
;
Hu, Chen
;
Wang, Haizhen
;
Liu, Jing
;
Wang, Wenchao
;
Liu, Qingsong
收藏
  |  
浏览/下载:76/0
  |  
提交时间:2022/01/25
A nanoselenium-coating biomimetic cytomembrane nanoplatform for mitochondrial targeted chemotherapy- and chemodynamic therapy through manganese and doxorubicin codelivery
期刊论文
JOURNAL OF NANOBIOTECHNOLOGY, 2021, 卷号: 19
作者:
Xiao, Jianmin
;
Yan, Miao
;
Zhou, Ke
;
Chen, Hui
;
Xu, Zhaowei
;
Gan, Yuehao
;
Hong, Biao
;
Tian, Geng
;
Qian, Junchao
;
Zhang, Guilong
;
Wu, Zhengyan
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2021/08/30
Cell membrane
Reactive oxygen species
Superoxide dismutase-1
Glutathione peroxidase 4
Dual-mode therapeutic pathways
Drug delivery system
Nanocrystal-loaded liposome for targeted delivery of poorly water-soluble antitumor drugs with high drug loading and stability towards efficient cancer therapy
期刊论文
INTERNATIONAL JOURNAL OF PHARMACEUTICS, 2021, 卷号: 599
作者:
Liang, Huamin
;
Zou, Fengming
;
Liu, Qingwang
;
Wang, Beilei
;
Fu, Liyi
;
Liang, Xiaofei
;
Liu, Jing
;
Liu, Qingsong
收藏
  |  
浏览/下载:53/0
  |  
提交时间:2021/05/17
Liposome
Drug nanocrystal
Core-shell
Drug delivery
Tumor therapy
BCR-ABL
Decline in serum progastrin-releasing peptide predicts the response of patients with small cell lung cancer to chemotherapy
期刊论文
ONCOLOGY LETTERS, 2020, 卷号: 20
作者:
Li, Ming
;
Han, Dandan
;
Wang, Wei
;
Zhang, Yang
;
Li, Dan
;
Dai, Chunyang
;
Qian, Liting
;
Lin, Wenchu
收藏
  |  
浏览/下载:49/0
  |  
提交时间:2020/12/28
progastrin-releasing peptide
therapeutic monitoring
small-cell lung cancer
neuron-specific enolase
Discovery of a highly potent and selective Bruton's tyrosine kinase inhibitor avoiding impairment of ADCC effects for B-cell non-Hodgkin lymphoma
期刊论文
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2020, 卷号: 5
作者:
Liu, Juan
;
Liang, Qianmao
;
Wang, Aoli
;
Zou, Fengming
;
Qi, Ziping
;
Yu, Kailin
;
Liu, Qingwang
;
Chen, Cheng
;
Liu, Jing
;
Liu, Qingsong
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2020/11/30
Osimertinib successfully combats EGFR-negative glioblastoma cells by inhibiting the MAPK pathway
期刊论文
ACTA PHARMACOLOGICA SINICA, 2020
作者:
Chen, Cheng
;
Cheng, Chuan-dong
;
Wu, Hong
;
Wang, Zuo-wei
;
Wang, Li
;
Jiang, Zong-ru
;
Wang, Ao-li
;
Hu, Chen
;
Dong, Yong-fei
;
Niu, Wan-xiang
;
Qi, Shuang
;
Qi, Zi-ping
;
Liu, Jing
;
Wang, Wen-chao
;
Niu, Chao-shi
;
Liu, Qing-song
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  |  
Adobe PDF(3476Kb)
  |  
收藏
  |  
浏览/下载:101/36
  |  
提交时间:2020/11/26
glioblastoma
osimertinib
temozolamide
MAPK-signaling pathway
MNK
eukaryotic translation initiation factor 4E
CRISPR/Cas9-related technologies in liver diseases: from feasibility to future diversity
期刊论文
INTERNATIONAL JOURNAL OF BIOLOGICAL SCIENCES, 2020, 卷号: 16
作者:
Xu, Ta
;
Li, Li
;
Liu, Yu-chen
;
Cao, Wei
;
Chen, Jia-si
;
Hu, Shuang
;
Liu, Ying
;
Li, Liang-yun
;
Zhou, Hong
;
Meng, Xiao-ming
;
Huang, Cheng
;
Zhang, Lei
;
Li, Jun
;
Zhou, Huan
收藏
  |  
浏览/下载:63/0
  |  
提交时间:2020/11/26
CRISPR/Cas9
viral hepatitis
hepatocellular carcinoma (HCC)
clinical research
Discovery of N-(4-(6-Acetamidopyrimidin-4-yloxy)phenyl)-2-(2-(trifluoromethyl)phenyl)acetamide (CHMFL-FLT3-335) as a Potent FMS-like Tyrosine Kinase 3 Internal Tandem Duplication (FLT3-ITD) Mutant Selective Inhibitor for Acute Myeloid Leukemia
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 2, 页码: 875-892
作者:
Liang, Xiaofei
;
Wang, Beilei
;
Chen, Cheng
;
Wang, Aoli
;
Hu, Chen
;
Zou, Fengming
;
Yu, Kailin
;
Liu, Qingwang
;
Li, Feng
;
Hu, Zhenquan
;
Lu, Tingting
;
Wang, Junjie
;
Wang, Li
;
Weisberg, Ellen L.
;
Li, Lili
;
Xia, Ruixiang
;
Wang, Wenchao
;
Ren, Tao
;
Ge, Jian
;
Liu, Jing
;
Liu, Qinsong
浏览
  |  
Adobe PDF(13868Kb)
  |  
收藏
  |  
浏览/下载:377/322
  |  
提交时间:2020/05/21
Sodium chloride (NaCl) potentiates digoxin-induced anti-tumor activity in small cell lung cancer
期刊论文
CANCER BIOLOGY & THERAPY, 2019, 卷号: 20, 期号: 1, 页码: 52-64
作者:
Deng, Ke
;
Shen, Jiawei
;
Wang, Wei
;
Li, Ming
;
Li, Hong
;
Chen, Cheng
;
Zhao, Huan
;
Zhang, Mei
;
Xue, Tian
;
Liu, Qingsong
;
Lui, Vivian Wai Yan
;
Hong, Bo
;
Lin, Wenchu
浏览
  |  
Adobe PDF(3554Kb)
  |  
收藏
  |  
浏览/下载:71/28
  |  
提交时间:2020/03/31
small cell lung cancer
digoxin
NaCl
cardiac glycosides
ATP1A1