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中国科学院合肥物质科学研究院机构知识库
Knowledge Management System of Hefei Institute of Physical Science,CAS
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Acetaldehyde induces similar cytotoxic and genotoxic risks in BEAS-2B cells and HHSteCs: involvement of differential regulation of MAPK/ERK and PI3K/AKT pathways
期刊论文
ENVIRONMENTAL SCIENCE AND POLLUTION RESEARCH, 2023, 卷号: 30
作者:
Zhang, Jingni
;
Wang, Hongjuan
;
Chen, Huan
;
Liu, Yong
;
Wang, An
;
Hou, Hongwei
;
Hu, Qingyuan
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浏览/下载:31/0
  |  
提交时间:2023/11/17
Acetaldehyde
Cytotoxicity
Genotoxicity
BEAS-2B cells
HHSteCs
MAPK/ERK
PI3K/AKT
Osimertinib successfully combats EGFR-negative glioblastoma cells by inhibiting the MAPK pathway
期刊论文
ACTA PHARMACOLOGICA SINICA, 2020
作者:
Chen, Cheng
;
Cheng, Chuan-dong
;
Wu, Hong
;
Wang, Zuo-wei
;
Wang, Li
;
Jiang, Zong-ru
;
Wang, Ao-li
;
Hu, Chen
;
Dong, Yong-fei
;
Niu, Wan-xiang
;
Qi, Shuang
;
Qi, Zi-ping
;
Liu, Jing
;
Wang, Wen-chao
;
Niu, Chao-shi
;
Liu, Qing-song
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Adobe PDF(3476Kb)
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浏览/下载:103/36
  |  
提交时间:2020/11/26
glioblastoma
osimertinib
temozolamide
MAPK-signaling pathway
MNK
eukaryotic translation initiation factor 4E
Discovery of 2-(4-Chloro-3-(trifluoromethyl)phenyl)-N-(4-((6,7-dimethoxyquinolin-4-yl)oxy)phenyl)acetamide (CHMFL-KIT-64) as a Novel Orally Available Potent Inhibitor against Broad-Spectrum Mutants of
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019
作者:
Yun Wu
;
Beilei Wang
;
Junjie Wang
;
Qi S(亓爽)
;
Fengming Zou
;
Ziping Qi
;
Feiyang Liu
;
Wenchao Wang
;
Qingsong Liu
;
Jing Liu
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Adobe PDF(5207Kb)
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浏览/下载:131/66
  |  
提交时间:2020/10/20
Transgenerational effects of diesel particulate matter on Caenorhabditis elegans through maternal and multigenerational exposure
期刊论文
ECOTOXICOLOGY AND ENVIRONMENTAL SAFETY, 2019, 卷号: 170, 期号: 无, 页码: 635-643
作者:
Wang, Mudi
;
Nie, Yaguang
;
Liu, Ying
;
Dai, Hui
;
Wang, Jingjing
;
Si, Bo
;
Yang, Zhen
;
Cheng, Lei
;
Liu, Yun
;
Chen, Shaopeng
;
Xu, An
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Adobe PDF(6386Kb)
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浏览/下载:127/45
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提交时间:2020/05/21
Diesel Particulate Matter
Caenorhabditis elegans
Multigenerational
Reproductive toxicity
Germ cell apoptosis
Nuclear factor (erythroid-derived 2)-like 2 antioxidative response mitigates cytoplasmic radiation-induced DNA double-strand breaks
期刊论文
CANCER SCIENCE, 2019, 卷号: 110, 期号: 2, 页码: 686-696
作者:
Wang, Jun
;
Konishi, Teruaki
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Adobe PDF(913Kb)
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浏览/下载:78/37
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提交时间:2020/05/21
cytoplasm
double-strand DNA break
mitochondria
radiation biology
Discovery of N-(4-(6-Acetamidopyrimidin-4-yloxy)phenyl)-2-(2-(trifluoromethyl)phenyl)acetamide (CHMFL-FLT3-335) as a Potent FMS-like Tyrosine Kinase 3 Internal Tandem Duplication (FLT3-ITD) Mutant Selective Inhibitor for Acute Myeloid Leukemia
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 2, 页码: 875-892
作者:
Liang, Xiaofei
;
Wang, Beilei
;
Chen, Cheng
;
Wang, Aoli
;
Hu, Chen
;
Zou, Fengming
;
Yu, Kailin
;
Liu, Qingwang
;
Li, Feng
;
Hu, Zhenquan
;
Lu, Tingting
;
Wang, Junjie
;
Wang, Li
;
Weisberg, Ellen L.
;
Li, Lili
;
Xia, Ruixiang
;
Wang, Wenchao
;
Ren, Tao
;
Ge, Jian
;
Liu, Jing
;
Liu, Qinsong
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Adobe PDF(13868Kb)
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浏览/下载:378/323
  |  
提交时间:2020/05/21
Discovery of (E)-N-(4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)-3-((3-(2-(pyridin-2-yl)vinyl)-1H-indazol-6-yl)thio)propanamide (CHMFL-ABL-121) as a highly potent ABL kinase inhibitor capable of overcoming a variety of ABL mutants including T315I for chronic myeloid leukemia
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 160, 页码: 61-81
作者:
Liu, Xuesong
;
Wang, Beilei
;
Chen, Cheng
;
Jiang, Zongru
;
Hu, Chen
;
Wu, Hong
;
Zhang, Yicong
;
Liu, Xiaochuan
;
Wang, Wenliang
;
Wang, Junjie
;
Hu, Zhenquan
;
Wang, Aoli
;
Huang, Tao
;
Liu, Qingwang
;
Wang, Wei
;
Wang, Li
;
Wang, Wenchao
;
Ren, Tao
;
Li, Lili
;
Xia, Ruixiang
;
Ge, Jian
;
Liu, Qingsong
;
Liu, Jing
Adobe PDF(4593Kb)
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浏览/下载:198/104
  |  
提交时间:2019/01/11
ABL kinase
Kinase inhibitor
ABL mutant
CML
Targeting Nrf2-mediated heme oxygenase-1 enhances non-thermal plasma-induced cell death in non-small-cell lung cancer A549 cells
期刊论文
ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS, 2018, 卷号: 658, 页码: 54-65
作者:
Ma, Jie
;
Yu, K. N.
;
Cheng, Cheng
;
Ni, Guohua
;
Shen, Jie
;
Han, Wei
Adobe PDF(4120Kb)
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浏览/下载:97/44
  |  
提交时间:2019/01/11
Non-thermal plasma
Reactive oxygen species
Heme oxygenase-1
Apoptotic death
c-JUN N-terminal kinase
N-acetylcysteine protects against microcystin-LR-induced endoplasmic reticulum stress and germ cell apoptosis in zebrafish testes
期刊论文
CHEMOSPHERE, 2018, 卷号: 204, 期号: 无, 页码: 463-473
作者:
Zhao, Sujuan
;
Liu, Ying
;
Wang, Fang
;
Xu, Dexiang
;
Xie, Ping
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Adobe PDF(4185Kb)
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浏览/下载:69/31
  |  
提交时间:2019/08/23
Microcystin
Endoplasmic reticulum stress
Apoptosis
N-acetylcysteine (NAC)
Zebrafish testes
Discovery of 4-((N-(2-(dimethylamino)ethyl)acrylamido)methyl)-N-(4-methyl-3-((4-(pyridin-3-yl)pyrimidin-2-yl)amino)phenyl)benzamide (CHMFL-PDGFR-159) as a highly selective type II PDGFR alpha kinase inhibitor for PDGFR alpha driving chronic eosinophilic leukemia
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 150, 期号: 无, 页码: 366-384
作者:
Wang, Qiang
;
Liu, Feiyang
;
Qi, Shuang
;
Qi, Ziping
;
Yan, Xiao-E.
;
Wang, Beilei
;
Wang, Aoli
;
Wang, Wei
;
Chen, Cheng
;
Liu, Xiaochuan
;
Jiang, Zongru
;
Hu, Zhenquan
;
Wang, Li
;
Wang, Wenchao
;
Ren, Tao
;
Zhang, Shanchun
;
Yun, Cai-Hong
;
Liu, Qingsong
;
Liu, Jing
浏览
  |  
Adobe PDF(5108Kb)
  |  
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浏览/下载:598/506
  |  
提交时间:2019/06/10
PDGFR kinase
Type II inhibitor
Kinase inhibitor
CEL