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中国科学院合肥物质科学研究院机构知识库
Knowledge Management System of Hefei Institute of Physical Science,CAS
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Nitrogen and boron dual-doped graphene quantum dots for near-infrared second window imaging and photothermal therapy
期刊论文
APPLIED MATERIALS TODAY, 2019, 卷号: 14, 期号: 无, 页码: 108-117
作者:
Wang, Hui
;
Mu, Qingxin
;
Wang, Kui
;
Revia, Richard A.
;
Yen, Charles
;
Gu, Xinyu
;
Tian, Bowei
;
Liu, Jun
;
Zhang, Miqin
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Adobe PDF(3141Kb)
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浏览/下载:1673/138
  |  
提交时间:2020/05/21
Theranostic nanoparticle
NIR II fluorescence imaging
Graphene quantum dot
Photothermal effect
Cancer therapy
Sodium chloride (NaCl) potentiates digoxin-induced anti-tumor activity in small cell lung cancer
期刊论文
CANCER BIOLOGY & THERAPY, 2019, 卷号: 20, 期号: 1, 页码: 52-64
作者:
Deng, Ke
;
Shen, Jiawei
;
Wang, Wei
;
Li, Ming
;
Li, Hong
;
Chen, Cheng
;
Zhao, Huan
;
Zhang, Mei
;
Xue, Tian
;
Liu, Qingsong
;
Lui, Vivian Wai Yan
;
Hong, Bo
;
Lin, Wenchu
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  |  
Adobe PDF(3554Kb)
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浏览/下载:71/28
  |  
提交时间:2020/03/31
small cell lung cancer
digoxin
NaCl
cardiac glycosides
ATP1A1
Discovery of 4-((N-(2-(dimethylamino)ethyl)acrylamido)methyl)-N-(4-methyl-3-((4-(pyridin-3-yl)pyrimidin-2-yl)amino)phenyl)benzamide (CHMFL-PDGFR-159) as a highly selective type II PDGFR alpha kinase inhibitor for PDGFR alpha driving chronic eosinophilic leukemia
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 150, 期号: 无, 页码: 366-384
作者:
Wang, Qiang
;
Liu, Feiyang
;
Qi, Shuang
;
Qi, Ziping
;
Yan, Xiao-E.
;
Wang, Beilei
;
Wang, Aoli
;
Wang, Wei
;
Chen, Cheng
;
Liu, Xiaochuan
;
Jiang, Zongru
;
Hu, Zhenquan
;
Wang, Li
;
Wang, Wenchao
;
Ren, Tao
;
Zhang, Shanchun
;
Yun, Cai-Hong
;
Liu, Qingsong
;
Liu, Jing
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Adobe PDF(5108Kb)
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浏览/下载:596/506
  |  
提交时间:2019/06/10
PDGFR kinase
Type II inhibitor
Kinase inhibitor
CEL
Magnetic field direction differentially impacts the growth of different cell types
期刊论文
ELECTROMAGNETIC BIOLOGY AND MEDICINE, 2018, 卷号: 37, 期号: 2, 页码: 114-125
作者:
Tian, Xiaofei
;
Wang, Dongmei
;
Zha, Meng
;
Yang, Xingxing
;
Ji, Xinmiao
;
Zhang, Lei
;
Zhang, Xin
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Adobe PDF(2690Kb)
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浏览/下载:186/52
  |  
提交时间:2019/08/26
Magnetic resonance imaging (MRI)
static magnetic field (SMF)
magnetic field direction
cancer cells
non-cancer cells
Identification of a selective and direct NLRP3 inhibitor to treat inflammatory disorders
期刊论文
JOURNAL OF EXPERIMENTAL MEDICINE, 2017, 卷号: 214, 期号: 11, 页码: 3219-3238
作者:
Jiang, Hua
;
He, Hongbin
;
Chen, Yun
;
Huang, Wei
;
Cheng, Jinbo
;
Ye, Jin
;
Wang, Aoli
;
Tao, Jinhui
;
Wang, Chao
;
Liu, Qingsong
;
Jin, Tengchuan
;
Jiang, Wei
;
Deng, Xianming
;
Zhou, Rongbin
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Adobe PDF(2740Kb)
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浏览/下载:230/160
  |  
提交时间:2019/06/17
Discovery and characterization of a novel irreversible EGFR mutants selective and potent kinase inhibitor CHMFL-EGFR-26 with a distinct binding mode
期刊论文
ONCOTARGET, 2017, 卷号: 8, 期号: 11, 页码: 18359-18372
作者:
Hu, Chen
;
Wang, Aoli
;
Wu, Hong
;
Qi, Ziping
;
Li, Xixiang
;
Yan, Xiao-E
;
Chen, Cheng
;
Yu, Kailin
;
Zou, Fengming
;
Wang, Wenchao
;
Wang, Wei
;
Wu, Jiaxin
;
Liu, Juan
;
Wang, Beilei
;
Wang, Li
;
Ren, Tao
;
Zhang, Shanchun
;
Yun, Cai-Hong
;
Liu, Jing
;
Liu, Qingsong
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  |  
Adobe PDF(6153Kb)
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浏览/下载:183/48
  |  
提交时间:2018/07/04
Egfr
Egfrt790m
Nsclc
Kinase Inhibitors
Drug Resistance
Rutin ameliorates obesity through brown fat activation
期刊论文
FASEB JOURNAL, 2017, 卷号: 31, 期号: 1, 页码: 333-+
作者:
Yuan, Xiaoxue
;
Wei, Gang
;
You, Yilin
;
Huang, Yuanyuan
;
Lee, Hyuek Jong
;
Dong, Meng
;
Lin, Jun
;
Hu, Tao
;
Zhang, Hanlin
;
Zhang, Chuanhai
;
Zhou, Huiqiao
;
Ye, Rongcai
;
Qi, Xiaolong
;
Zhai, Baiqiang
;
Huang, Weidong
;
Liu, Shunai
;
Xie, Wen
;
Liu, Qingsong
;
Liu, Xiaomeng
;
Cui, Chengbi
;
Li, Donghao
;
Zhan, Jicheng
;
Cheng, Jun
;
Yuan, Zengqiang
;
Jin, Wanzhu
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  |  
Adobe PDF(2063Kb)
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浏览/下载:164/45
  |  
提交时间:2018/07/04
Brown Adipose Tissue
Rutin
Obesity
Energy Expenditure
Mitochondria
Simultaneous inhibition of Vps34 kinase would enhance PI3K delta inhibitor cytotoxicity in the B-cell malignancies
期刊论文
ONCOTARGET, 2016, 卷号: 7, 期号: 33, 页码: 53515-53525
作者:
Liu, Xiaochuan
;
Wang, Aoli
;
Liang, Xiaofei
;
Liu, Juanjuan
;
Zou, Fengming
;
Chen, Cheng
;
Zhao, Zheng
;
Deng, Yuanxin
;
Wu, Hong
;
Qi, Ziping
;
Wang, Beilei
;
Wang, Li
;
Liu, Feiyang
;
Xu, Yunhe
;
Wang, Wenchao
;
Fernandes, Stacey M.
;
Stone, Richard M.
;
Galinsky, Ilene A.
;
Brown, Jennifer R.
;
Loh, Teckpeng
;
Griffin, James. D.
;
Zhang, Shanchun
;
Weisberg, Ellen L.
;
Zhang, Xin
;
Liu, Jing
;
Liu, Qingsong
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  |  
Adobe PDF(7625Kb)
  |  
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  |  
浏览/下载:100/38
  |  
提交时间:2017/11/21
Pi3k Delta
Vps34
Combination
Chronic Lymphatic Leukemia
Acute Myeloid Leukemia
Discovery and characterization of a novel potent type II native and mutant BCR-ABL inhibitor (CHMFL-074) for Chronic Myeloid Leukemia (CML)
期刊论文
ONCOTARGET, 2016, 卷号: 7, 期号: 29, 页码: 45562-45574
作者:
Liu, Feiyang
;
Wang, Beilei
;
Wang, Qiang
;
Qi, Ziping
;
Chen, Cheng
;
Kong, Lu-Lu
;
Chen, Ji-Yun
;
Liu, Xiaochuan
;
Wang, Aoli
;
Hu, Chen
;
Wang, Wenchao
;
Wang, Huiping
;
Wu, Fan
;
Ruan, Yanjie
;
Qi, Shuang
;
Liu, Juan
;
Zou, Fengming
;
Hu, Zhenquan
;
Wang, Wei
;
Wang, Li
;
Zhang, Shanchun
;
Yun, Cai-Hong
;
Zhai, Zhimin
;
Liu, Jing
;
Liu, Qingsong
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  |  
Adobe PDF(8054Kb)
  |  
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  |  
浏览/下载:254/200
  |  
提交时间:2017/11/21
Bcr-abl
Pdgfr
Chronic Myeloid Leukemia
Kinase Inhibitor
Discovery of N-(34(1-lsonicotinoylpiperidin-4-yl)oxy)-4methylpheny1)-3-(trifluoromethyl)benzamide (CHMFL-KIT-110) as a Selective, Potent, and Orally Available Type II c-KIT Kinase Inhibitor for Gastrointestinal Stromal Tumors (GISTs)
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 8, 页码: 3964-3979
作者:
Wang, Qang
;
Liu, Feiyang
;
Wang, Beilei
;
Zou, Fengming
;
Chen, Cheng
;
Liu, Xiaochuan
;
Wang, Aoli
;
Qi, Shuang
;
Wang, Wenchao
;
Qi, Ziping
;
Zhao, Zheng
;
Hu, Zhenquan
;
Wang, Wei
;
Wang, Li
;
Zhang, Shanchun
;
Wang, Yuexiang
;
Liu, Jing
;
Liu, Qingsong
浏览
  |  
Adobe PDF(10221Kb)
  |  
收藏
  |  
浏览/下载:128/75
  |  
提交时间:2017/11/10