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Discovery and characterization of a novel highly potent and selective type II native and drug-resistant V299L mutant BCR-ABL inhibitor (CHMFL-ABL-039) for Chronic Myeloid Leukemia (CML) 期刊论文
CANCER BIOLOGY & THERAPY, 2019, 卷号: 20, 期号: 6, 页码: 877-885
作者:  Wu, Jiaxin;  Wang, Aoli;  Li, Xixiang;  Chen, Cheng;  Qi, Ziping;  Hu, Chen;  Wang, Wenliang;  Wu, Hong;  Huang, Tao;  Zhao, Ming;  Wang, Wenchao;  Hu, Zhenquan;  Liu, Qingwang;  Wang, Beilei;  Wang, Li;  Li, Lili;  Ge, Jian;  Ren, Tao;  Xia, Ruixiang;  Liu, Jing
收藏  |  浏览/下载:59/0  |  提交时间:2019/11/27
BCR-ABL  PDGFR  chronic myeloid leukemia  kinase inhibitor  
Giant antiferromagnetic negative thermal expansion in (MnNiGe)(1-x)(MnCoSn)(x) compounds 期刊论文
JOURNAL OF ALLOYS AND COMPOUNDS, 2019, 卷号: 782, 期号: 无, 页码: 881-886
作者:  Zhu, Feng;  Lin, Jianchao;  Zhang, Xuekai;  Li, Longfu;  Yang, Cheng;  Wang, Meng;  Wu, Ying;  Tong, Peng;  Song, Wenhai;  Sun, Yuping
浏览  |  Adobe PDF(2150Kb)  |  收藏  |  浏览/下载:93/41  |  提交时间:2020/05/21
Negative thermal expansion  Martensitic transformation  AFM ground state  Magnetostriction  Thermal conductivity  
Discovery of N-(4-(6-Acetamidopyrimidin-4-yloxy)phenyl)-2-(2-(trifluoromethyl)phenyl)acetamide (CHMFL-FLT3-335) as a Potent FMS-like Tyrosine Kinase 3 Internal Tandem Duplication (FLT3-ITD) Mutant Selective Inhibitor for Acute Myeloid Leukemia 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 2, 页码: 875-892
作者:  Liang, Xiaofei;  Wang, Beilei;  Chen, Cheng;  Wang, Aoli;  Hu, Chen;  Zou, Fengming;  Yu, Kailin;  Liu, Qingwang;  Li, Feng;  Hu, Zhenquan;  Lu, Tingting;  Wang, Junjie;  Wang, Li;  Weisberg, Ellen L.;  Li, Lili;  Xia, Ruixiang;  Wang, Wenchao;  Ren, Tao;  Ge, Jian;  Liu, Jing;  Liu, Qinsong
浏览  |  Adobe PDF(13868Kb)  |  收藏  |  浏览/下载:378/323  |  提交时间:2020/05/21
Dual Graphitic-N Doping in a Six-Membered C-Ring of Graphene-Analogous Particles Enables an Efficient Electrocatalyst for the Hydrogen Evolution Reaction 期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2019
作者:  Lin, Zhiyu;  Yang, Yang;  Li, Mengsi;  Huang, Hao;  Hu, Wei;  Cheng, Ling;  Yan, Wensheng;  Yu, Zhiwu;  Mao, Kaitian;  Xia, Guoliang;  Lu, Jian;  Jiang, Peng;  ang, Kang;  Zhang, Ruirui;  Xu, Pengping;  Wang, Changlai;  Hu, Lin;  Chen, Qianwang
浏览  |  Adobe PDF(5160Kb)  |  收藏  |  浏览/下载:80/36  |  提交时间:2020/10/29
Discovery of (E)-N-(4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)-3-((3-(2-(pyridin-2-yl)vinyl)-1H-indazol-6-yl)thio)propanamide (CHMFL-ABL-121) as a highly potent ABL kinase inhibitor capable of overcoming a variety of ABL mutants including T315I for chronic myeloid leukemia 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 160, 页码: 61-81
作者:  Liu, Xuesong;  Wang, Beilei;  Chen, Cheng;  Jiang, Zongru;  Hu, Chen;  Wu, Hong;  Zhang, Yicong;  Liu, Xiaochuan;  Wang, Wenliang;  Wang, Junjie;  Hu, Zhenquan;  Wang, Aoli;  Huang, Tao;  Liu, Qingwang;  Wang, Wei;  Wang, Li;  Wang, Wenchao;  Ren, Tao;  Li, Lili;  Xia, Ruixiang;  Ge, Jian;  Liu, Qingsong;  Liu, Jing
Adobe PDF(4593Kb)  |  收藏  |  浏览/下载:198/104  |  提交时间:2019/01/11
ABL kinase  Kinase inhibitor  ABL mutant  CML  
Isotropic Low Thermal Expansion over a Wide Temperature Range in Ti1-xZrxF3+x (0.1 <= x <= 0.5) Solid Solutions 期刊论文
INORGANIC CHEMISTRY, 2018, 卷号: 57, 期号: 22, 页码: 14396-14400
作者:  Yang, Cheng;  Zhang, Yugang;  Bai, Jianming;  Tong, Peng;  Lin, Jianchao;  Tong, Haiyun;  Zhang, Lei;  Wen, Wen;  Zhang, Xingmin;  Sun, Yuping
收藏  |  浏览/下载:37/0  |  提交时间:2019/12/25
Enhanced mechanical properties and large magnetocaloric effect in epoxy-bonded Mn0.98CoGe 期刊论文
SCRIPTA MATERIALIA, 2018, 卷号: 150, 期号: 无, 页码: 96-100
作者:  Zhu, F.;  Lin, J. C.;  Jiang, W. B.;  Yang, C.;  Li, L. F.;  Zhang, X. K.;  Song, W. H.;  Zhu, X. B.;  Tong, P.;  Sun, Y. P.
浏览  |  Adobe PDF(1356Kb)  |  收藏  |  浏览/下载:108/63  |  提交时间:2019/08/23
First-order magnetic phase transition  Mechanical properties  Magnetocaloric effect  Relative cooling powder  Thermal conductivity  
Acceleration of Kirkendall effect processes in silicon nanospheres using magnetic fields 期刊论文
CrystEngComm, 2018, 卷号: 20, 期号: 6, 页码: 710-715
作者:  Yuecheng Bian;  Wei Ding;  Lin Hu;  Zongwei Ma;  Long Cheng;  Ranran Zhang;  Xuebin Zhu;  Xianwu Tang;  Jianming Dai;  Jin Bai;  Yuping Sun;  Zhigao Sheng
浏览  |  Adobe PDF(1801Kb)  |  收藏  |  浏览/下载:108/50  |  提交时间:2018/10/18
Discovery of 1-(4-(4-Amino-3-(4-(2-morpholinoethoxy)-phenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)phenyl)-3-(5-(tert-butyl)isoxazol-3-yl)urea (CHMFL-FLT3-213) as a Highly Potent Type II FLT3 Kinase Inhibitor Capable of Overcoming a Variety of FLT3 Kinase Mutants in FLT3-ITD Positive AML 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 20, 页码: 8407-8424
作者:  Wang, Aoli;  Li, Xixiang;  Chen, Cheng;  Wu, Hong;  Qi, Ziping;  Hu, Chen;  Yu, Kailin;  Wu, Jiaxin;  Liu, Juan;  Liu, Xiaochuan;  Hu, Zhenquan;  Wang, Wei;  Wang, Wenliang;  Wang, Wenchao;  Wang, Li;  Wang, Beilei;  Liu, Qingwang;  Li, Lili;  Ge, Jian;  Ren, Tao;  Zhang, Shanchun;  Xia, Ruixiang;  Liu, Jing;  Liu, Qingsong
浏览  |  Adobe PDF(10028Kb)  |  收藏  |  浏览/下载:86/31  |  提交时间:2019/06/17
Colossal negative thermal expansion with an extended temperature interval covering room temperature in fine-powdered Mn0.98CoGe 期刊论文
APPLIED PHYSICS LETTERS, 2016, 卷号: 109, 期号: 24, 页码: 241903
作者:  Lin, Jianchao;  Tong, Peng;  Zhang, Kui;  Tong, Haiyun;  Guo, Xinge;  Yang, Cheng;  Wu, Ying;  Wang, Meng;  Lin, Shuai;  Chen, Li;  Song, Wenhai;  Sun, Yuping
浏览  |  Adobe PDF(2005Kb)  |  收藏  |  浏览/下载:147/66  |  提交时间:2017/09/12