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中国科学院合肥物质科学研究院机构知识库
Knowledge Management System of Hefei Institute of Physical Science,CAS
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Predicting and overcoming resistance to CDK9 inhibitors for cancer therapy
期刊论文
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13
作者:
Hua, Chen
;
Shena, Lijuan
;
Zoua, Fengming
;
Wua, Yun
;
Wanga, Beilei
;
Wanga, Aoli
;
Wud, Chao
;
Wanga, Li
;
Liua, Jing
;
Wanga, Wenchao
;
Liua, Qingsong
收藏
  |  
浏览/下载:43/0
  |  
提交时间:2023/11/10
Acquired resistance mutations
CDK9 inhibitors
Transcription
Single nucleotide polymorphisms
BAY1251152
Discovery of Pyrrolo[2,3-d]pyrimidine derivatives as potent and selective colony stimulating factor 1 receptor kinase inhibitors
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 243
作者:
Liang, Xiaofei
;
Wang, Chun
;
Wang, Beilei
;
Liu, Juan
;
Qi, Shuang
;
Wang, Aoli
;
Liu, Qingwang
;
Deng, Maoqing
;
Wang, Li
;
Liu, Jing
;
Liu, Qingsong
收藏
  |  
浏览/下载:45/0
  |  
提交时间:2022/12/23
CSF1R inhibitor
Kinase inhibitor
Macrophage polarization
Repurposing of the FGFR inhibitor AZD4547 as a potent inhibitor of necroptosis by selectively targeting RIPK1
期刊论文
ACTA PHARMACOLOGICA SINICA, 2022
作者:
Wang, Zuo-wei
;
Zou, Feng-ming
;
Wang, Ao-li
;
Yang, Jing
;
Jin, Rui
;
Wang, Bei-lei
;
Shen, Li-juan
;
Qi, Shuang
;
Liu, Juan
;
Liu, Jing
;
Wang, Wen-chao
;
Liu, Qing-song
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2022/12/22
AZD4547
RIPK1
inhibitors
SIRS model
anti-necroptosis
A spiropyran with low pK(a) for tracking DNA G-quadruplexes and revealing the dissipation of Delta Psi m with senescence using an in-situ switching strategy
期刊论文
SENSORS AND ACTUATORS B-CHEMICAL, 2022, 卷号: 359
作者:
Tian, Xinrong
;
Li, Jin
;
Zhang, Yanhui
;
Gao, Ying
;
Afzal, Muhammad Wasim
;
Wang, Aoli
;
James, Tony D.
;
Bai, Yinjuan
;
Guo, Yuan
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2022/12/22
Fluorescent probes
G-quadruplexes
Membrane potential of mitochondria
Senescence
Senescent cells
CHMFL-26 is a highly potent irreversible HER2 inhibitor for use in the treatment of HER2-positive and HER2-mutant cancers
期刊论文
ACTA PHARMACOLOGICA SINICA, 2022
作者:
Cao, Jiang-yan
;
Qi, Shuang
;
Wu, Hong
;
Wang, Ao-li
;
Liu, Qing-wang
;
Li, Xi-xiang
;
Wang, Bei-lei
;
Ge, Juan
;
Zou, Feng-ming
;
Chen, Cheng
;
Wang, Jun-jie
;
Hu, Chen
;
Liu, Jing
;
Wang, Wen-chao
;
Liu, Qing-song
收藏
  |  
浏览/下载:106/0
  |  
提交时间:2022/03/28
HER2
breast cancers
gastric cancers
irreversible inhibitor
drug resistance
Inhibition of the deubiquitinating enzyme USP47 as a novel targeted therapy for hematologic malignancies expressing mutant EZH2
期刊论文
LEUKEMIA, 2022
作者:
Yang, Jing
;
Weisberg, Ellen L.
;
Qi, Shuang
;
Ni, Wei
;
Mei, Husheng
;
Wang, Zuowei
;
Meng, Chengcheng
;
Zhang, Shengzhe
;
Hou, Mingqi
;
Qi, Ziping
;
Wang, Aoli
;
Jiang, Yunyun
;
Jiang, Zongru
;
Huang, Tao
;
Liu, Qingwang
;
Magin, Robert S.
;
Doherty, Laura
;
Wang, Wenchao
;
Liu, Jing
;
Buhrlage, Sara J.
;
Liu, Qingsong
;
Griffin, James D.
收藏
  |  
浏览/下载:84/0
  |  
提交时间:2022/02/14
Targeting chaperon protein HSP70 as a novel therapeutic strategy for FLT3-ITD-positive acute myeloid leukemia
期刊论文
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2021, 卷号: 6
作者:
Hu, Chen
;
Zou, Fengming
;
Wang, Aoli
;
Miao, Weili
;
Liang, Qianmao
;
Weisberg, Ellen L.
;
Wang, Yinsheng
;
Liu, Jing
;
Wang, Wenchao
;
Liu, Qingsong
收藏
  |  
浏览/下载:64/0
  |  
提交时间:2021/11/01
Discovery of a highly potent kinase inhibitor capable of overcoming multiple imatinib-resistant ABL mutants for chronic myeloid leukemia (CML)
期刊论文
EUROPEAN JOURNAL OF PHARMACOLOGY, 2021, 卷号: 897
作者:
Lu, Tingting
;
Cao, Jiangyan
;
Zou, Fengming
;
Li, Xixiang
;
Wang, Aoli
;
Wang, Wenliang
;
Liang, Huamin
;
Liu, Qingwang
;
Hu, Chen
;
Chen, Cheng
;
Hu, Zhenquan
;
Wang, Wenchao
;
Li, Lili
;
Ge, Jian
;
Shen, Yang
;
Ren, Tao
;
Liu, Jing
;
Xia, Ruixiang
;
Liu, Qingsong
收藏
  |  
浏览/下载:86/0
  |  
提交时间:2021/04/26
BCR-ABL
ABL mutants
Chronic myeloid leukemia
Kinase inhibitor
Imatinib resistance
Selectively targeting FLT3-ITD mutants over FLT3-wt by a novel inhibitor for acute myeloid leukemia
期刊论文
HAEMATOLOGICA, 2021, 卷号: 106
作者:
Wang, Aoli
;
Hu, Chen
;
Chen, Cheng
;
Liang, Xiaofei
;
Wang, Beilei
;
Zou, Fengming
;
Yu, Kailin
;
Li, Feng
;
Liu, Qingwang
;
Qi, Ziping
;
Wang, Junjie
;
Wang, Wenliang
;
Wang, Li
;
Weisberg, Ellen L.
;
Wang, Wenchao
;
Li, Lili
;
Ge, Jian
;
Xia, Ruixiang
;
Liu, Jing
;
Liu, Qingsong
收藏
  |  
浏览/下载:57/0
  |  
提交时间:2021/04/26
Discovery of a highly potent and selective Bruton's tyrosine kinase inhibitor avoiding impairment of ADCC effects for B-cell non-Hodgkin lymphoma
期刊论文
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2020, 卷号: 5
作者:
Liu, Juan
;
Liang, Qianmao
;
Wang, Aoli
;
Zou, Fengming
;
Qi, Ziping
;
Yu, Kailin
;
Liu, Qingwang
;
Chen, Cheng
;
Liu, Jing
;
Liu, Qingsong
收藏
  |  
浏览/下载:53/0
  |  
提交时间:2020/11/30