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Discovery and characterization of a novel highly potent and selective type II native and drug-resistant V299L mutant BCR-ABL inhibitor (CHMFL-ABL-039) for Chronic Myeloid Leukemia (CML) 期刊论文
CANCER BIOLOGY & THERAPY, 2019, 卷号: 20, 期号: 6, 页码: 877-885
作者:  Wu, Jiaxin;  Wang, Aoli;  Li, Xixiang;  Chen, Cheng;  Qi, Ziping;  Hu, Chen;  Wang, Wenliang;  Wu, Hong;  Huang, Tao;  Zhao, Ming;  Wang, Wenchao;  Hu, Zhenquan;  Liu, Qingwang;  Wang, Beilei;  Wang, Li;  Li, Lili;  Ge, Jian;  Ren, Tao;  Xia, Ruixiang;  Liu, Jing
收藏  |  浏览/下载:59/0  |  提交时间:2019/11/27
BCR-ABL  PDGFR  chronic myeloid leukemia  kinase inhibitor  
Increase of Co 3d projected electronic density of states in AgCoO2 enabled an efficient electrocatalyst toward oxygen evolution reaction 期刊论文
NANO ENERGY, 2019, 卷号: 57, 期号: 无, 页码: 753-760
作者:  Zhang, Ruirui;  Sun, Zhongti;  Zong, Cichang;  Lin, Zhiyu;  Huang, Hao;  Yang, Kang;  Chen, Jing;  Liu, Shuai;  Huang, Minxue;  Yang, Yang;  Zhang, Wenhua;  Chen, Qianwang
浏览  |  Adobe PDF(5751Kb)  |  收藏  |  浏览/下载:82/42  |  提交时间:2020/05/21
AgCoO2  Interfacial charge transfer state  AgCoO2/Ag hybrid  Surface charge states  OER  Theory calculations  
Improvement of Cr (VI) photoreduction under visible-light by g-C3N4 modified by nano-network structured palygorskite 期刊论文
CHEMICAL ENGINEERING JOURNAL, 2019, 卷号: 358, 页码: 398-407
作者:  Zhang, Jing;  Gao, Ning;  Chen, Fulong;  Zhang, Tao;  Zhang, Guilong;  Wang, Dongfang;  Xie, Xingyong;  Cai, Dongqing;  Ma, Xijun;  Wu, Lifang;  Wu, Zhengyan
Adobe PDF(2784Kb)  |  收藏  |  浏览/下载:191/56  |  提交时间:2019/01/09
Palygorskite  Graphitic carbon nitride  Ion beam bombardment  Photocatalysts  
Discovery of N-(4-(6-Acetamidopyrimidin-4-yloxy)phenyl)-2-(2-(trifluoromethyl)phenyl)acetamide (CHMFL-FLT3-335) as a Potent FMS-like Tyrosine Kinase 3 Internal Tandem Duplication (FLT3-ITD) Mutant Selective Inhibitor for Acute Myeloid Leukemia 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 2, 页码: 875-892
作者:  Liang, Xiaofei;  Wang, Beilei;  Chen, Cheng;  Wang, Aoli;  Hu, Chen;  Zou, Fengming;  Yu, Kailin;  Liu, Qingwang;  Li, Feng;  Hu, Zhenquan;  Lu, Tingting;  Wang, Junjie;  Wang, Li;  Weisberg, Ellen L.;  Li, Lili;  Xia, Ruixiang;  Wang, Wenchao;  Ren, Tao;  Ge, Jian;  Liu, Jing;  Liu, Qinsong
浏览  |  Adobe PDF(13868Kb)  |  收藏  |  浏览/下载:378/323  |  提交时间:2020/05/21
Repurposing cabozantinib to GISTs: Overcoming multiple imatinib-resistant cKIT mutations including gatekeeper and activation loop mutants in GISTs preclinical models 期刊论文
CANCER LETTERS, 2019, 页码: 105-114
作者:  Lu, Tingting;  Chen, Cheng;  Wang, Aoli;  Jiang, Zongru;  Qi, Ziping;  Hu, Zhenquan;  Hu, Chen;  Liu, Feiyang;  Wang, Wenliang;  Wu, Hong;  Wang, Beilei;  Wang, Li;  Qi, Shuang;  Wu, Jiaxin;  Wang, Wenchao;  Tang, Jun;  Yan, Hezhong;  Bai, Mingfeng;  Liu, Qingsong;  Liu, Jing
收藏  |  浏览/下载:28/0  |  提交时间:2020/07/14
cKIT T670I mutant  Activation loop mutants  Drug resistance  
Magnetic field-induced electronic phase transition in the Dirac semimetal state of black phosphorus under pressure 期刊论文
SCIENCE BULLETIN, 2018, 卷号: 63, 期号: 23, 页码: 1539-1544
作者:  Sun, Zeliang;  Xiang, Ziji;  Wang, Zhongyi;  Zhang, Jinglei;  Ma, Long;  Wang, Naizhou;  Shang, Chao;  Meng, Fanbao;  Zou, Liangjian;  Zhang, Yuanbo;  Chen, Xianhui
收藏  |  浏览/下载:37/0  |  提交时间:2019/12/25
Black phosphorus  High magnetic field  Quantum limit  Electron phase transition  
Origin of the structural phase transition in single-crystal TaTe2 期刊论文
PHYSICAL REVIEW B, 2018, 卷号: 98, 期号: 22, 页码: 7
作者:  Gao, J. J.;  Si, J. G.;  Luo, X.;  Yan, J.;  Chen, F. C.;  Lin, G. T.;  Hu, L.;  Zhang, R. R.;  Tong, P.;  Song, W. H.;  Zhu, X. B.;  Lu, W. J.;  Sun, Y. P.
收藏  |  浏览/下载:48/0  |  提交时间:2019/12/25
Discovery of (E)-N-(4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)-3-((3-(2-(pyridin-2-yl)vinyl)-1H-indazol-6-yl)thio)propanamide (CHMFL-ABL-121) as a highly potent ABL kinase inhibitor capable of overcoming a variety of ABL mutants including T315I for chronic myeloid leukemia 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 160, 页码: 61-81
作者:  Liu, Xuesong;  Wang, Beilei;  Chen, Cheng;  Jiang, Zongru;  Hu, Chen;  Wu, Hong;  Zhang, Yicong;  Liu, Xiaochuan;  Wang, Wenliang;  Wang, Junjie;  Hu, Zhenquan;  Wang, Aoli;  Huang, Tao;  Liu, Qingwang;  Wang, Wei;  Wang, Li;  Wang, Wenchao;  Ren, Tao;  Li, Lili;  Xia, Ruixiang;  Ge, Jian;  Liu, Qingsong;  Liu, Jing
Adobe PDF(4593Kb)  |  收藏  |  浏览/下载:198/104  |  提交时间:2019/01/11
ABL kinase  Kinase inhibitor  ABL mutant  CML  
Refreshing Piezoelectrics: Distinctive Role of Manganese in Lead Free Perovskites 期刊论文
ACS APPLIED MATERIALS & INTERFACES, 2018, 卷号: 10, 期号: 43, 页码: 37298-37306
作者:  Yao, Fang-Zhou;  Zhang, Mao-Hua;  Wang, Ke;  Zhou, Jia-Jun;  Chen, Feng;  Xu, Bin;  Li, Fei;  Shen, Yang;  Zhang, Qing-Hua;  Gu, Lin;  Zhang, Xiao-Wen;  Li, Jing-Feng
Adobe PDF(2258Kb)  |  收藏  |  浏览/下载:99/41  |  提交时间:2019/01/09
(K,Na)NbO3  lead free  perovskite  piezoelectric  manganese doping  
Discovery of 4-(((4-(5-chloro-2-(((1s,4s)-4-((2-methoxyethyl)amino) cyclohexyl)amino)pyridin-4-yl)thiazol-2-yl)amino)methyl) tetrahydro-2H-pyran-4-carbonitrile (JSH-150) as a novel highly selective and potent CDK9 kinase inhibitor 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 158, 页码: 896-916
作者:  Wang, Beilei;  Wu, Jiaxin;  Wu, Yun;  Chen, Cheng;  Zou, Fengming;  Wang, Aoli;  Wu, Hong;  Hu, Zhenquan;  Jiang, Zongru;  Liu, Qingwang;  Wang, Wei;  Zhang, Yicong;  Liu, Feiyang;  Zhao, Ming;  Hu, Jie;  Huang, Tao;  Ge, Juan;  Wang, Li;  Ren, Tao;  Wang, Yuxin;  Liu, Jing;  Liu, Qingsong
收藏  |  浏览/下载:29/0  |  提交时间:2019/12/25
CDK9  Kinase inhibitor  Structure-activity relationship  Leukemia