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中国科学院合肥物质科学研究院机构知识库
Knowledge Management System of Hefei Institute of Physical Science,CAS
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收录类别:SCI
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WOS被引频次降序
Discovery and characterization of a novel highly potent and selective type II native and drug-resistant V299L mutant BCR-ABL inhibitor (CHMFL-ABL-039) for Chronic Myeloid Leukemia (CML)
期刊论文
CANCER BIOLOGY & THERAPY, 2019, 卷号: 20, 期号: 6, 页码: 877-885
作者:
Wu, Jiaxin
;
Wang, Aoli
;
Li, Xixiang
;
Chen, Cheng
;
Qi, Ziping
;
Hu, Chen
;
Wang, Wenliang
;
Wu, Hong
;
Huang, Tao
;
Zhao, Ming
;
Wang, Wenchao
;
Hu, Zhenquan
;
Liu, Qingwang
;
Wang, Beilei
;
Wang, Li
;
Li, Lili
;
Ge, Jian
;
Ren, Tao
;
Xia, Ruixiang
;
Liu, Jing
收藏
  |  
浏览/下载:52/0
  |  
提交时间:2019/11/27
BCR-ABL
PDGFR
chronic myeloid leukemia
kinase inhibitor
Discovery of (E)-N-(4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)-3-((3-(2-(pyridin-2-yl)vinyl)-1H-indazol-6-yl)thio)propanamide (CHMFL-ABL-121) as a highly potent ABL kinase inhibitor capable of overcoming a variety of ABL mutants including T315I for chronic myeloid leukemia
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 160, 页码: 61-81
作者:
Liu, Xuesong
;
Wang, Beilei
;
Chen, Cheng
;
Jiang, Zongru
;
Hu, Chen
;
Wu, Hong
;
Zhang, Yicong
;
Liu, Xiaochuan
;
Wang, Wenliang
;
Wang, Junjie
;
Hu, Zhenquan
;
Wang, Aoli
;
Huang, Tao
;
Liu, Qingwang
;
Wang, Wei
;
Wang, Li
;
Wang, Wenchao
;
Ren, Tao
;
Li, Lili
;
Xia, Ruixiang
;
Ge, Jian
;
Liu, Qingsong
;
Liu, Jing
Adobe PDF(4593Kb)
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  |  
浏览/下载:191/104
  |  
提交时间:2019/01/11
ABL kinase
Kinase inhibitor
ABL mutant
CML
Discovery of 4-((N-(2-(dimethylamino)ethyl)acrylamido)methyl)-N-(4-methyl-3-((4-(pyridin-3-yl)pyrimidin-2-yl)amino)phenyl)benzamide (CHMFL-PDGFR-159) as a highly selective type II PDGFR alpha kinase inhibitor for PDGFR alpha driving chronic eosinophilic leukemia
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 150, 期号: 无, 页码: 366-384
作者:
Wang, Qiang
;
Liu, Feiyang
;
Qi, Shuang
;
Qi, Ziping
;
Yan, Xiao-E.
;
Wang, Beilei
;
Wang, Aoli
;
Wang, Wei
;
Chen, Cheng
;
Liu, Xiaochuan
;
Jiang, Zongru
;
Hu, Zhenquan
;
Wang, Li
;
Wang, Wenchao
;
Ren, Tao
;
Zhang, Shanchun
;
Yun, Cai-Hong
;
Liu, Qingsong
;
Liu, Jing
浏览
  |  
Adobe PDF(5108Kb)
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  |  
浏览/下载:589/505
  |  
提交时间:2019/06/10
PDGFR kinase
Type II inhibitor
Kinase inhibitor
CEL
c-Abl inhibition mitigates diet-induced obesity through improving insulin sensitivity of subcutaneous fat in mice
期刊论文
DIABETOLOGIA, 2017, 卷号: 60, 期号: 5, 页码: 900-910
作者:
Wu, Rong
;
Sun, Jian-guang
;
Wang, Ji-qiu
;
Li, Binhua
;
Liu, Qingsong
;
Ning, Guang
;
Jin, Wanzhu
;
Yuan, Zengqiang
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2018/07/26
Discovery of 2-((3-Acrylamido-4-methylphenyl)amino)-N-(2-methyl5-(3,4,5-trimethoxybenzamido)phenyI)-4-(methylamino)pyrimidine-5-carboxamide (CHMFL-BMX-078) as a Highly Potent and Selective Type II Irreversible Bone Marrow Kinase in the X Chromosome (BMX) Kinase Inhibitor
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 5, 页码: 1793-1816
作者:
Liang, Xiaofei
;
Lv, Fengchao
;
Wang, Beilei
;
Yu, Kailin
;
Wu, Hong
;
Qi, Ziping
;
Jiang, Zongru
;
Chen, Cheng
;
Wang, Aoli
;
Miao, Weili
;
Wang, Wenchao
;
Hu, Zhenquan
;
Liu, Juan
;
Liu, Xiaochuan
;
Zhao, Zheng
;
Wang, Li
;
Zhang, Shanchuan
;
Ye, Zi
;
Wang, Chu
;
Ren, Tao
;
Wang, Yinsheng
;
Liu, Qingsong
;
Liu, Jing
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  |  
Adobe PDF(5919Kb)
  |  
收藏
  |  
浏览/下载:17294/7523
  |  
提交时间:2018/07/04
Discovery of 4-Methyl-N-(44(4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)-3-((1-nicotinoylpiperidin-4-y1)oxy)benzamide (CHMFL-ABL/KIT-155) as a Novel Highly Potent Type II ABL/KIT Dual Kinase Inhibitor with a Distinct Hinge Binding
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 1, 页码: 273-289
作者:
Wang, Qiang
;
Liu, Feiyang
;
Wang, Beilei
;
Zou, Fengming
;
Qi, Ziping
;
Chen, Cheng
;
Yu, Kailin
;
Hu, Chen
;
Qi, Shuang
;
Wang, Wenchao
;
Hu, Zhenquan
;
Liu, Juan
;
Wang, Wei
;
Wang, Li
;
Liang, Qianmao
;
Zhang, Shanchun
;
Ren, Tao
;
Liu, Qingsong
;
Liu, Jing
浏览
  |  
Adobe PDF(3516Kb)
  |  
收藏
  |  
浏览/下载:101/58
  |  
提交时间:2018/07/04
Discovery of N-((1-(4-(3-(3-((6,7-Dimethoxyquinolin-3-yl)oxy)phenyl)ureido)-2-(trifluoromethyl)phenyl)piperidin-4-yl)methyl)propionamide (CHMFL-KIT-8140) as a Highly Potent Type II Inhibitor Capable of Inhibiting the T670I "Gatekeeper" Mutant of cKIT Kinase
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 18, 页码: 8456-8472
作者:
Li, Binhua
;
Wang, Aoli
;
Liu, Juan
;
Qi, Ziping
;
Liu, Xiaochuan
;
Yu, Kailin
;
Wu, Hong
;
Chen, Cheng
;
Hu, Chen
;
Wang, Wenchao
;
Wu, Jiaxin
;
Hu, Zhenquan
;
Ye, Ling
;
Zou, Fengming
;
Liu, Feiyang
;
Wang, Beilei
;
Wang, Li
;
Ren, Tao
;
Zhang, Shaojuan
;
Bai, Mingfeng
;
Zhang, Shanchun
;
Liu, Jing
;
Liu, Qingsong
浏览
  |  
Adobe PDF(2856Kb)
  |  
收藏
  |  
浏览/下载:1402/1298
  |  
提交时间:2017/11/21
Discovery and characterization of a novel potent type II native and mutant BCR-ABL inhibitor (CHMFL-074) for Chronic Myeloid Leukemia (CML)
期刊论文
ONCOTARGET, 2016, 卷号: 7, 期号: 29, 页码: 45562-45574
作者:
Liu, Feiyang
;
Wang, Beilei
;
Wang, Qiang
;
Qi, Ziping
;
Chen, Cheng
;
Kong, Lu-Lu
;
Chen, Ji-Yun
;
Liu, Xiaochuan
;
Wang, Aoli
;
Hu, Chen
;
Wang, Wenchao
;
Wang, Huiping
;
Wu, Fan
;
Ruan, Yanjie
;
Qi, Shuang
;
Liu, Juan
;
Zou, Fengming
;
Hu, Zhenquan
;
Wang, Wei
;
Wang, Li
;
Zhang, Shanchun
;
Yun, Cai-Hong
;
Zhai, Zhimin
;
Liu, Jing
;
Liu, Qingsong
浏览
  |  
Adobe PDF(8054Kb)
  |  
收藏
  |  
浏览/下载:247/196
  |  
提交时间:2017/11/21
Bcr-abl
Pdgfr
Chronic Myeloid Leukemia
Kinase Inhibitor
Dual Inhibition of AKT/FLT3-ITD by A674563 Overcomes FLT3 Ligand-Induced Drug Resistance in FLT3-ITD positive AML
期刊论文
ONCOTARGET, 2016, 卷号: 7, 期号: 20, 页码: 29131-29142
作者:
Wang, Aoli
;
Wu, Hong
;
Chen, Cheng
;
Hu, Chen
;
Qi, Ziping
;
Wang, Wenchao
;
Yu, Kailin
;
Liu, Xiaochuan
;
Zou, Fengming
;
Zhao, Zheng
;
Wu, Jiaxin
;
Liu, Juan
;
Liu, Feiyang
;
Wang, Li
;
Stone, Richard M.
;
Galinksy, Ilene A.
;
Griffin, James D.
;
Zhang, Shanchun
;
Weisberg, Ellen L.
;
Liu, Jing
;
Liu, Qingsong
浏览
  |  
Adobe PDF(4786Kb)
  |  
收藏
  |  
浏览/下载:132/35
  |  
提交时间:2017/11/16
Acute Myeloid Leukemia
Flt3-itd
Akt
A6745763
Flt3-ligand
Discovery of N-(34(1-lsonicotinoylpiperidin-4-yl)oxy)-4methylpheny1)-3-(trifluoromethyl)benzamide (CHMFL-KIT-110) as a Selective, Potent, and Orally Available Type II c-KIT Kinase Inhibitor for Gastrointestinal Stromal Tumors (GISTs)
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 8, 页码: 3964-3979
作者:
Wang, Qang
;
Liu, Feiyang
;
Wang, Beilei
;
Zou, Fengming
;
Chen, Cheng
;
Liu, Xiaochuan
;
Wang, Aoli
;
Qi, Shuang
;
Wang, Wenchao
;
Qi, Ziping
;
Zhao, Zheng
;
Hu, Zhenquan
;
Wang, Wei
;
Wang, Li
;
Zhang, Shanchun
;
Wang, Yuexiang
;
Liu, Jing
;
Liu, Qingsong
浏览
  |  
Adobe PDF(10221Kb)
  |  
收藏
  |  
浏览/下载:123/72
  |  
提交时间:2017/11/10