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中国科学院合肥物质科学研究院机构知识库
Knowledge Management System of Hefei Institute of Physical Science,CAS
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Zanubrutinib monotherapy for relapsed or refractory non-germinal center diffuse large B-cell lymphoma
期刊论文
BLOOD ADVANCES, 2022, 卷号: 6
作者:
Yang, Haiyan
;
Xiang, Bing
;
Song, Yuqin
;
Zhang, Huilai
;
Zhao, Weili
;
Zou, Dehui
;
Lv, Fangfang
;
Guo, Wei
;
Liu, Aichun
;
Li, Caixia
;
Tan, Ziwen
;
Liu, Yang
;
Fu, Lina
;
Guo, Haiyi
;
Novotny, William
;
Huang, Jane
;
Li, Yufu
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2022/12/23
Characterization of the metabolites of tirabrutinib generated from rat, dog and human liver microsomes using ultra-high-performance liquid chromatography combined with high-resolution mass spectrometry
期刊论文
RAPID COMMUNICATIONS IN MASS SPECTROMETRY, 2022, 卷号: 36
作者:
Zhang, Hongjian
;
Hu, Zhen
;
Zhang, Huiping
;
Sun, Xiyan
;
Yang, Jianming
;
Yuan, Jie
收藏
  |  
浏览/下载:48/0
  |  
提交时间:2022/03/28
Bruton's tyrosine kinase inhibitors in primary central nervous system lymphoma-evaluation of anti-tumor efficacy and brain distribution
期刊论文
TRANSLATIONAL CANCER RESEARCH, 2021, 卷号: 10
作者:
Yu, Haifeng
;
Kong, Haiying
;
Li, Cong
;
Dong, Xiaowu
;
Wu, Yizhe
;
Zhuang, Yuxin
;
Han, Shuiyun
;
Lei, Tao
;
Yang, Haiyan
收藏
  |  
浏览/下载:52/0
  |  
提交时间:2021/08/31
Primary central nervous system lymphoma ( PCNSL)
Bruton's tyrosine kinase (BTK)
ibrutinib
zanubrutinib
tirabrutinib
Discovery of 4,7-Diamino-5-(4-phenoxyphenyl)-6-methylene-pyrinnido[5,4-b]pyrrolizines as Novel Bruton's Tyrosine Kinase Inhibitors
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 10, 页码: 4608-4627
作者:
Xue, Yu
;
Song, Peiran
;
Song, Zilan
;
Wang, Aoli
;
Tong, Linjiang
;
Geng, Meiyu
;
Ding, Jian
;
Liu, Qingsong
;
Sun, Liping
;
Xie, Hua
;
Zhang, Ao
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Adobe PDF(6587Kb)
  |  
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  |  
浏览/下载:147/106
  |  
提交时间:2019/08/23
Venetoclax and low-dose cytarabine induced complete remission in a patient with high-risk acute myeloid leukemia: a case report
期刊论文
FRONTIERS OF MEDICINE, 2018, 卷号: 12
-
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浏览/下载:24/0
  |  
提交时间:2020/10/26
BCL-2 INHIBITOR
MIDOSTAURIN
CLASSIFICATION
DECITABINE
MECHANISMS
MUTATIONS
TARGETS
IDH
BTK
venetoclax
cytarabine
AML
leukemia
Discovery of 1-(4-(4-Amino-3-(4-(2-morpholinoethoxy)-phenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)phenyl)-3-(5-(tert-butyl)isoxazol-3-yl)urea (CHMFL-FLT3-213) as a Highly Potent Type II FLT3 Kinase Inhibitor Capable of Overcoming a Variety of FLT3 Kinase Mutants in FLT3-ITD Positive AML
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 20, 页码: 8407-8424
作者:
Wang, Aoli
;
Li, Xixiang
;
Chen, Cheng
;
Wu, Hong
;
Qi, Ziping
;
Hu, Chen
;
Yu, Kailin
;
Wu, Jiaxin
;
Liu, Juan
;
Liu, Xiaochuan
;
Hu, Zhenquan
;
Wang, Wei
;
Wang, Wenliang
;
Wang, Wenchao
;
Wang, Li
;
Wang, Beilei
;
Liu, Qingwang
;
Li, Lili
;
Ge, Jian
;
Ren, Tao
;
Zhang, Shanchun
;
Xia, Ruixiang
;
Liu, Jing
;
Liu, Qingsong
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  |  
Adobe PDF(10028Kb)
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  |  
浏览/下载:78/31
  |  
提交时间:2019/06/17
Structure-activity relationship investigation for benzonaphthyridinone derivatives as novel potent Bruton's tyrosine kinase (BTK) irreversible inhibitors
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 137, 页码: 545-557
作者:
Wang, Beilei
;
Deng, Yuanxin
;
Chen, Yongfei
;
Yu, Kailin
;
Wang, Aoli
;
Liang, Qianmao
;
Wang, Wei
;
Chen, Cheng
;
Wu, Hong
;
Hu, Chen
;
Miao, Weili
;
Hur, Wooyoung
;
Wang, Wenchao
;
Hu, Zhenquan
;
Weisberg, Ellen L.
;
Wang, Jinhua
;
Ren, Tao
;
Wang, Yinsheng
;
Gray, Nathanael S.
;
Liu, Qingsong
;
Liu, Jing
收藏
  |  
浏览/下载:347/0
  |  
提交时间:2018/08/16
Btk
Kinase Inhibitor
Irreversible Inhibitor
Structure-activity Relationship
B-cell Lymphoma
Discovery of N-(3-(5-((3-acrylamido-4-(morpholine-4-carbonyl) phenyl)amino)-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-methylphenyl)-4-(tert-butyl)benzamide (CHMFL-BTK-01) as a highly selective irreversible Bruton's tyrosine kinase (BTK) inhibitor
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 131, 页码: 107-125
作者:
Liang, Qianmao
;
Chen, Yongfei
;
Yu, Kailin
;
Chen, Cheng
;
Zhang, Shouxiang
;
Wang, Aoli
;
Wang, Wei
;
Wu, Hong
;
Liu, Xiaochuan
;
Wang, Beilei
;
Wang, Li
;
Hu, Zhenquan
;
Wang, Wenchao
;
Ren, Tao
;
Zhang, Shanchun
;
Liu, Qingsong
;
Yun, Cai-Hong
;
Liu, Jing
收藏
  |  
浏览/下载:47/0
  |  
提交时间:2018/07/26
Btk
Irreversible Inhibitor
Kinase Inhibitor
Structure-activity Relationship
B-cell Lymphoma
Irreversible inhibition of BTK kinase by a novel highly selective inhibitor CHMFL-BTK-11 suppresses inflammatory response in rheumatoid arthritis model
期刊论文
SCIENTIFIC REPORTS, 2017, 卷号: 7, 期号: 无, 页码: 1-10
作者:
Wu, Hong
;
Huang, Qiong
;
Qi, Ziping
;
Chen, Yongfei
;
Wang, Aoli
;
Chen, Cheng
;
Liang, Qianmao
;
Wang, Jinghua
;
Chen, Wensheng
;
Dong, Jin
;
Yu, Kailin
;
Hu, Chen
;
Wang, Wenchao
;
Liu, Xiaochuan
;
Deng, Yuanxin
;
Wang, Li
;
Wang, Beilei
;
Li, Xiaoxiang
;
Gray, Nathanael S.
;
Liu, Jing
;
Wei, Wei
;
Liu, Qingsong
浏览
  |  
Adobe PDF(3966Kb)
  |  
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  |  
浏览/下载:121/63
  |  
提交时间:2018/07/04
Discovery of 2-((3-Acrylamido-4-methylphenyl)amino)-N-(2-methyl5-(3,4,5-trimethoxybenzamido)phenyI)-4-(methylamino)pyrimidine-5-carboxamide (CHMFL-BMX-078) as a Highly Potent and Selective Type II Irreversible Bone Marrow Kinase in the X Chromosome (BMX) Kinase Inhibitor
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 5, 页码: 1793-1816
作者:
Liang, Xiaofei
;
Lv, Fengchao
;
Wang, Beilei
;
Yu, Kailin
;
Wu, Hong
;
Qi, Ziping
;
Jiang, Zongru
;
Chen, Cheng
;
Wang, Aoli
;
Miao, Weili
;
Wang, Wenchao
;
Hu, Zhenquan
;
Liu, Juan
;
Liu, Xiaochuan
;
Zhao, Zheng
;
Wang, Li
;
Zhang, Shanchuan
;
Ye, Zi
;
Wang, Chu
;
Ren, Tao
;
Wang, Yinsheng
;
Liu, Qingsong
;
Liu, Jing
浏览
  |  
Adobe PDF(5919Kb)
  |  
收藏
  |  
浏览/下载:17293/7523
  |  
提交时间:2018/07/04