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中国科学院合肥物质科学研究院机构知识库
Knowledge Management System of Hefei Institute of Physical Science,CAS
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Predicting and overcoming resistance to CDK9 inhibitors for cancer therapy
期刊论文
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13
作者:
Hua, Chen
;
Shena, Lijuan
;
Zoua, Fengming
;
Wua, Yun
;
Wanga, Beilei
;
Wanga, Aoli
;
Wud, Chao
;
Wanga, Li
;
Liua, Jing
;
Wanga, Wenchao
;
Liua, Qingsong
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2023/11/10
Acquired resistance mutations
CDK9 inhibitors
Transcription
Single nucleotide polymorphisms
BAY1251152
Discovery of Pyrrolo[2,3-d]pyrimidine derivatives as potent and selective colony stimulating factor 1 receptor kinase inhibitors
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 243
作者:
Liang, Xiaofei
;
Wang, Chun
;
Wang, Beilei
;
Liu, Juan
;
Qi, Shuang
;
Wang, Aoli
;
Liu, Qingwang
;
Deng, Maoqing
;
Wang, Li
;
Liu, Jing
;
Liu, Qingsong
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2022/12/23
CSF1R inhibitor
Kinase inhibitor
Macrophage polarization
Pulmonary Salivary Gland Tumor, Mucoepidermoid Carcinoma: A Literature Review
期刊论文
JOURNAL OF ONCOLOGY, 2022, 卷号: 2022
作者:
Hu, Shumin
;
Gong, Jiali
;
Zhu, Xiu
;
Lu, Hongyang
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2022/12/23
Repurposing of the FGFR inhibitor AZD4547 as a potent inhibitor of necroptosis by selectively targeting RIPK1
期刊论文
ACTA PHARMACOLOGICA SINICA, 2022
作者:
Wang, Zuo-wei
;
Zou, Feng-ming
;
Wang, Ao-li
;
Yang, Jing
;
Jin, Rui
;
Wang, Bei-lei
;
Shen, Li-juan
;
Qi, Shuang
;
Liu, Juan
;
Liu, Jing
;
Wang, Wen-chao
;
Liu, Qing-song
收藏
  |  
浏览/下载:45/0
  |  
提交时间:2022/12/22
AZD4547
RIPK1
inhibitors
SIRS model
anti-necroptosis
E3 ubiquitin ligase NEDD4L negatively regulates inflammation by promoting ubiquitination of MEKK2
期刊论文
EMBO REPORTS, 2022
作者:
Li, Hui
;
Wang, Ning
;
Jiang, Yu
;
Wang, Haofei
;
Xin, Zengfeng
;
An, Huazhang
;
Pan, Hao
;
Ma, Wangqian
;
Zhang, Ting
;
Wang, Xiaojian
;
Lin, Wenlong
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2022/12/22
IL-17R signaling
inflammation
MEKK2
NEDD4L
ubiquitination
Expert consensus on the diagnosis and treatment of NTRK gene fusion solid tumors in China
期刊论文
THORACIC CANCER, 2022
作者:
Xu, Chunwei
;
Si, Lu
;
Wang, Wenxian
;
Li, Ziming
;
Song, Zhengbo
;
Wang, Qian
;
Liu, Aijun
;
Yu, Jinpu
;
Fang, Wenfeng
;
Zhong, Wenzhao
;
Wang, Zhijie
;
Zhang, Yongchang
;
Liu, Jingjing
;
Zhang, Shirong
;
Cai, Xiuyu
;
Liu, Anwen
;
Li, Wen
;
Zhan, Ping
;
Liu, Hongbing
;
Lv, Tangfeng
;
Miao, Liyun
;
Min, Lingfeng
;
Chen, Yu
;
Yuan, Jingping
;
Wang, Feng
;
Jiang, Zhansheng
;
Lin, Gen
;
Pu, Xingxiang
;
Lin, Rongbo
;
Liu, Weifeng
;
Rao, Chuangzhou
;
Lv, Dongqing
;
Yu, Zongyang
;
Lei, Lei
;
Li, Xiaoyan
;
Tang, Chuanhao
;
Zhou, Chengzhi
;
Zhang, Junping
;
Xue, Junli
;
Guo, Hui
;
Chu, Qian
;
Meng, Rui
;
Wu, Jingxun
;
Zhang, Rui
;
Hu, Xiao
;
Zhou, Jin
;
Zhu, Zhengfei
;
Li, Yongheng
;
Qiu, Hong
;
Xia, Fan
;
Lu, Yuanyuan
;
Chen, Xiaofeng
;
Ge, Rui
;
Dai, Enyong
;
Han, Yu
;
Pan, Weiwei
;
Luo, Jiancheng
;
Jia, Hongtao
;
Dong, Xiaowei
;
Pang, Fei
;
Wang, Kai
;
Wang, Liping
;
Zhu, Youcai
;
Xie, Yanru
;
Lin, Xinqin
;
Cai, Jing
;
Wei, Jia
;
Lan, Fen
;
Feng, Huijing
;
Wang, Lin
;
Du, Yingying
;
Yao, Wang
;
Shi, Xuefei
;
Niu, Xiaomin
;
Yuan, Dongmei
;
Yao, Yanwen
;
Huang, Jianhui
;
Zhang, Yinbin
;
Sun, Pingli
;
Wang, Hong
;
Ye, Mingxiang
;
Wang, Dong
;
Wang, Zhaofeng
;
Wan, Bing
;
Lv, Donglai
;
Wei, Qing
;
Kang, Jin
;
Zhang, Jiatao
;
Zhang, Chao
;
Yu, Genhua
;
Ou, Juanjuan
;
Shi, Lin
;
Li, Zhongwu
;
Liu, Zhefeng
;
Liu, Jing
;
Yang, Nong
;
Wu, Lin
;
Wang, Huijuan
;
Jin, Gu
;
Yang, Liu
;
Wang, Guansong
;
Fang, Meiyu
;
Fang, Yong
;
Li, Yuan
;
Wang, Xiaojia
;
Zhang, Yiping
;
Ma, Shenglin
;
Wang, Biyun
;
Zhang, Xiaotian
;
Song, Yong
;
Lu, Yuanzhi
收藏
  |  
浏览/下载:44/0
  |  
提交时间:2022/12/22
fusion
precision medicine
solid tumor
targeted therapy
tyrosine receptor kinase
CircVAPA promotes small cell lung cancer progression by modulating the miR-377-3p and miR-494-3p/IGF1R/AKT axis
期刊论文
Molecular Cancer, 2022, 卷号: 21
作者:
Hua,Jinghan
;
Wang,Xiaolin
;
Ma,Liying
;
Li,Jingxin
;
Cao,Guozhen
;
Zhang,Shaobo
;
Lin,Wenchu
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2022/12/22
CircVAPA
SCLC
Progression
miR-377-3p
miR-494-3p
IGF1R
AKT
BMS-536924
Systemic Therapy for Hepatocellular Carcinoma: Chinese Consensus-Based Interdisciplinary Expert Statements
期刊论文
LIVER CANCER, 2022, 卷号: 11
作者:
Sun, Yongkun
;
Zhang, Wen
;
Bi, Xinyu
;
Yang, Zhengqiang
;
Tang, Yu
;
Jiang, Liming
;
Bi, Feng
;
Chen, Minshan
;
Cheng, Shuqun
;
Chi, Yihebali
;
Han, Yue
;
Huang, Jing
;
Huang, Zhen
;
Ji, Yuan
;
Jia, Liqun
;
Jiang, Zhichao
;
Jin, Jing
;
Jin, Zhengyu
;
Li, Xiao
;
Li, Zhiyu
;
Liang, Jun
;
Liu, Lianxin
;
Liu, Yunpeng
;
Lu, Yinying
;
Lu, Shichun
;
Meng, Qinghua
;
Niu, Zuoxing
;
Pan, Hongming
;
Qin, Shukui
;
Qu, Wang
;
Shao, Guoliang
;
Shen, Feng
;
Song, Tianqiang
;
Song, Yan
;
Tao, Kaishan
;
Tian, Aiping
;
Wang, Jianhua
;
Wang, Wenling
;
Wang, Zhe
;
Wu, Liqun
;
Xia, Feng
;
Xing, Baocai
;
Xu, Jianming
;
Xue, Huadan
;
Yan, Dong
;
Yang, Lin
;
Ying, Jianming
;
Yun, Jingping
;
Zeng, Zhaochong
;
Zhang, Xuewen
;
Zhang, Yanqiao
;
Zhang, Yefan
;
Zhao, Jianjun
;
Zhou, Jianguo
;
Zhu, Xu
;
Zou, Yinghua
;
Dong, Jiahong
;
Fan, Jia
;
Lau, Wan Yee
;
Sun, Yan
;
Yu, Jinming
;
Zhao, Hong
;
Zhou, Aiping
;
Cai, Jianqiang
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2022/12/23
Chinese interdisciplinary experts
Hepatocellular carcinoma
Molecular targeted therapy
Consensus
Efficacy and safety of anlotinib with and without EGFR-TKIs or immunotherapy in the treatment of elder patients with non-small-cell lung cancer: a retrospective study
期刊论文
BMC PULMONARY MEDICINE, 2022, 卷号: 22
作者:
Wang, Wenxian
;
Shao, Lan
;
Xu, Yibing
;
Song, Zhengbo
;
Lou, Guangyuan
;
Zhang, Yiping
;
Chen, Ming
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2022/12/23
Non-small cell lung cancer
Prognosis
Angiogenesis
Tyrosine kinase inhibitors
Treatment outcomes and prognosis of patients with primary and acquired BRAF-mutated non-small cell lung cancer: A multicenter retrospective study
期刊论文
GENES CHROMOSOMES & CANCER, 2022
作者:
Wang, Wenxian
;
Gu, Xiaodong
;
Si, Jinfei
;
Pu, Xingxiang
;
Wang, Liping
;
Chen, Huafei
;
Xu, Chunwei
;
Zhang, Xiaoyan
;
Yuan, Hongling
;
Lou, Guangyuan
;
Shao, Lan
;
Zhang, Gu
;
Song, Zhengbo
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2022/05/16
BRAF mutation
immune checkpoint inhibitors
non-small cell lung cancer
PD-L1
targeted therapy