×
验证码:
换一张
忘记密码?
记住我
切换中国科技网通行证登录
×
切换中国科技网通行证登录
登录
中文版
|
English
中国科学院合肥物质科学研究院机构知识库
Knowledge Management System of Hefei Institute of Physical Science,CAS
登录
注册
ALL
ORCID
题名
作者
学科领域
关键词
文献类型
出处
收录类别
出版者
发表日期
存缴日期
资助项目
学科门类
学习讨论厅
图片搜索
粘贴图片网址
首页
研究单元&专题
作者
文献类型
学科分类
知识图谱
新闻&公告
在结果中检索
研究单元&专题
中科院强磁场科学中心 [9]
合肥创新院 [1]
医学 [1]
作者
刘青松 [10]
王傲莉 [10]
王文超 [9]
刘小川 [6]
胡晨 [6]
齐紫平 [6]
更多...
发表日期
2019 [1]
2018 [4]
2017 [2]
2016 [3]
语种
英语 [9]
出处
JOURNAL OF... [5]
EUROPEAN J... [4]
ONCOTARGET [1]
资助项目
National N... [3]
National N... [3]
Natural Sc... [3]
Frontier S... [2]
Hundred Ta... [2]
National K... [2]
更多...
资助机构
China "Tho... [3]
Chinese Ac... [3]
"Hundred T... [2]
CAS/SAFEA [2]
Frontier S... [2]
National N... [2]
更多...
收录类别
SCI [10]
摘要
文献类型
期刊论文 [10]
×
知识图谱
HFCAS OpenIR
开始提交
已提交作品
待认领作品
已认领作品
未提交全文
收藏管理
QQ客服
官方微博
反馈留言
(本次检索基于用户作品认领结果)
浏览/检索结果:
共10条,第1-10条
帮助
限定条件
作者:王傲莉
第一作者
已选(
0
)
清除
条数/页:
5
10
15
20
25
30
35
40
45
50
55
60
65
70
75
80
85
90
95
100
排序方式:
请选择
发表日期升序
发表日期降序
WOS被引频次升序
WOS被引频次降序
提交时间升序
提交时间降序
题名升序
题名降序
作者升序
作者降序
期刊影响因子升序
期刊影响因子降序
Discovery of N-(4-(6-Acetamidopyrimidin-4-yloxy)phenyl)-2-(2-(trifluoromethyl)phenyl)acetamide (CHMFL-FLT3-335) as a Potent FMS-like Tyrosine Kinase 3 Internal Tandem Duplication (FLT3-ITD) Mutant Selective Inhibitor for Acute Myeloid Leukemia
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 2, 页码: 875-892
作者:
Liang, Xiaofei
;
Wang, Beilei
;
Chen, Cheng
;
Wang, Aoli
;
Hu, Chen
;
Zou, Fengming
;
Yu, Kailin
;
Liu, Qingwang
;
Li, Feng
;
Hu, Zhenquan
;
Lu, Tingting
;
Wang, Junjie
;
Wang, Li
;
Weisberg, Ellen L.
;
Li, Lili
;
Xia, Ruixiang
;
Wang, Wenchao
;
Ren, Tao
;
Ge, Jian
;
Liu, Jing
;
Liu, Qinsong
浏览
  |  
Adobe PDF(13868Kb)
  |  
收藏
  |  
浏览/下载:369/319
  |  
提交时间:2020/05/21
Discovery of (E)-N-(4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)-3-((3-(2-(pyridin-2-yl)vinyl)-1H-indazol-6-yl)thio)propanamide (CHMFL-ABL-121) as a highly potent ABL kinase inhibitor capable of overcoming a variety of ABL mutants including T315I for chronic myeloid leukemia
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 160, 页码: 61-81
作者:
Liu, Xuesong
;
Wang, Beilei
;
Chen, Cheng
;
Jiang, Zongru
;
Hu, Chen
;
Wu, Hong
;
Zhang, Yicong
;
Liu, Xiaochuan
;
Wang, Wenliang
;
Wang, Junjie
;
Hu, Zhenquan
;
Wang, Aoli
;
Huang, Tao
;
Liu, Qingwang
;
Wang, Wei
;
Wang, Li
;
Wang, Wenchao
;
Ren, Tao
;
Li, Lili
;
Xia, Ruixiang
;
Ge, Jian
;
Liu, Qingsong
;
Liu, Jing
Adobe PDF(4593Kb)
  |  
收藏
  |  
浏览/下载:190/104
  |  
提交时间:2019/01/11
ABL kinase
Kinase inhibitor
ABL mutant
CML
Discovery of 4,7-Diamino-5-(4-phenoxyphenyl)-6-methylene-pyrinnido[5,4-b]pyrrolizines as Novel Bruton's Tyrosine Kinase Inhibitors
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 10, 页码: 4608-4627
作者:
Xue, Yu
;
Song, Peiran
;
Song, Zilan
;
Wang, Aoli
;
Tong, Linjiang
;
Geng, Meiyu
;
Ding, Jian
;
Liu, Qingsong
;
Sun, Liping
;
Xie, Hua
;
Zhang, Ao
浏览
  |  
Adobe PDF(6587Kb)
  |  
收藏
  |  
浏览/下载:147/106
  |  
提交时间:2019/08/23
Discovery of 4-((N-(2-(dimethylamino)ethyl)acrylamido)methyl)-N-(4-methyl-3-((4-(pyridin-3-yl)pyrimidin-2-yl)amino)phenyl)benzamide (CHMFL-PDGFR-159) as a highly selective type II PDGFR alpha kinase inhibitor for PDGFR alpha driving chronic eosinophilic leukemia
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 150, 期号: 无, 页码: 366-384
作者:
Wang, Qiang
;
Liu, Feiyang
;
Qi, Shuang
;
Qi, Ziping
;
Yan, Xiao-E.
;
Wang, Beilei
;
Wang, Aoli
;
Wang, Wei
;
Chen, Cheng
;
Liu, Xiaochuan
;
Jiang, Zongru
;
Hu, Zhenquan
;
Wang, Li
;
Wang, Wenchao
;
Ren, Tao
;
Zhang, Shanchun
;
Yun, Cai-Hong
;
Liu, Qingsong
;
Liu, Jing
浏览
  |  
Adobe PDF(5108Kb)
  |  
收藏
  |  
浏览/下载:589/505
  |  
提交时间:2019/06/10
PDGFR kinase
Type II inhibitor
Kinase inhibitor
CEL
Discovery of 4-((N-(2-(dimethylamino)ethyl)acrylamido)methyl)-N-(4-methyl-3-((4-(pyridin-3-yl)pyrimidin-2-yl)amino)phenyl)benzamide (CHMFL-PDGFR-159) as a highly selective type II PDGFRα kinase inhibi
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018
作者:
Qiang Wang
;
Feiyang Liu
;
Qi S(亓爽)
;
Ziping Qi
;
Beilei Wang
;
Aoli Wang
;
Zongru Jiang
;
Wenchao Wang
;
Qingsong Liu
;
Jing Liu
浏览
  |  
Adobe PDF(5108Kb)
  |  
收藏
  |  
浏览/下载:124/51
  |  
提交时间:2020/10/20
Discovery of 1-(4-(4-Amino-3-(4-(2-morpholinoethoxy)-phenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)phenyl)-3-(5-(tert-butyl)isoxazol-3-yl)urea (CHMFL-FLT3-213) as a Highly Potent Type II FLT3 Kinase Inhibitor Capable of Overcoming a Variety of FLT3 Kinase Mutants in FLT3-ITD Positive AML
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 20, 页码: 8407-8424
作者:
Wang, Aoli
;
Li, Xixiang
;
Chen, Cheng
;
Wu, Hong
;
Qi, Ziping
;
Hu, Chen
;
Yu, Kailin
;
Wu, Jiaxin
;
Liu, Juan
;
Liu, Xiaochuan
;
Hu, Zhenquan
;
Wang, Wei
;
Wang, Wenliang
;
Wang, Wenchao
;
Wang, Li
;
Wang, Beilei
;
Liu, Qingwang
;
Li, Lili
;
Ge, Jian
;
Ren, Tao
;
Zhang, Shanchun
;
Xia, Ruixiang
;
Liu, Jing
;
Liu, Qingsong
浏览
  |  
Adobe PDF(10028Kb)
  |  
收藏
  |  
浏览/下载:78/31
  |  
提交时间:2019/06/17
Discovery of N-(5-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)-4-methoxy-2-(4-methyl-1,4-diazepan-1-yl)phenyl)acrylamide (CHMFL-ALK/EGFR-050) as a potent ALK/EGFR dual kinase inhibitor capable of overcoming a variety of ALK/EGFR associated drug resistant mutants in NSCLC
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 139, 期号: 无, 页码: 674-697
作者:
Chen, Yongfei
;
Wu, Jiaxin
;
Wang, Aoli
;
Qi, Ziping
;
Jiang, Taoshan
;
Chen, Cheng
;
Zou, Fengming
;
Hu, Chen
;
Wang, Wei
;
Wu, Hong
;
Hu, Zhenquan
;
Wang, Wenchao
;
Wang, Beilei
;
Wang, Li
;
Ren, Tao
;
Zhang, Shanchun
;
Liu, Qingsong
;
Liu, Jing
浏览
  |  
Adobe PDF(12656Kb)
  |  
收藏
  |  
浏览/下载:21275/11466
  |  
提交时间:2018/08/17
Egfr
Alk
Dual Kinase Inhibitor
Non-small Cell Lung Cancer
Discovery of N-((1-(4-(3-(3-((6,7-Dimethoxyquinolin-3-yl)oxy)phenyl)ureido)-2-(trifluoromethyl)phenyl)piperidin-4-yl)methyl)propionamide (CHMFL-KIT-8140) as a Highly Potent Type II Inhibitor Capable of Inhibiting the T670I "Gatekeeper" Mutant of cKIT Kinase
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 18, 页码: 8456-8472
作者:
Li, Binhua
;
Wang, Aoli
;
Liu, Juan
;
Qi, Ziping
;
Liu, Xiaochuan
;
Yu, Kailin
;
Wu, Hong
;
Chen, Cheng
;
Hu, Chen
;
Wang, Wenchao
;
Wu, Jiaxin
;
Hu, Zhenquan
;
Ye, Ling
;
Zou, Fengming
;
Liu, Feiyang
;
Wang, Beilei
;
Wang, Li
;
Ren, Tao
;
Zhang, Shaojuan
;
Bai, Mingfeng
;
Zhang, Shanchun
;
Liu, Jing
;
Liu, Qingsong
浏览
  |  
Adobe PDF(2856Kb)
  |  
收藏
  |  
浏览/下载:1401/1298
  |  
提交时间:2017/11/21
Dual Inhibition of AKT/FLT3-ITD by A674563 Overcomes FLT3 Ligand-Induced Drug Resistance in FLT3-ITD positive AML
期刊论文
ONCOTARGET, 2016, 卷号: 7, 期号: 20, 页码: 29131-29142
作者:
Wang, Aoli
;
Wu, Hong
;
Chen, Cheng
;
Hu, Chen
;
Qi, Ziping
;
Wang, Wenchao
;
Yu, Kailin
;
Liu, Xiaochuan
;
Zou, Fengming
;
Zhao, Zheng
;
Wu, Jiaxin
;
Liu, Juan
;
Liu, Feiyang
;
Wang, Li
;
Stone, Richard M.
;
Galinksy, Ilene A.
;
Griffin, James D.
;
Zhang, Shanchun
;
Weisberg, Ellen L.
;
Liu, Jing
;
Liu, Qingsong
浏览
  |  
Adobe PDF(4786Kb)
  |  
收藏
  |  
浏览/下载:132/35
  |  
提交时间:2017/11/16
Acute Myeloid Leukemia
Flt3-itd
Akt
A6745763
Flt3-ligand
Discovery of N-(34(1-lsonicotinoylpiperidin-4-yl)oxy)-4methylpheny1)-3-(trifluoromethyl)benzamide (CHMFL-KIT-110) as a Selective, Potent, and Orally Available Type II c-KIT Kinase Inhibitor for Gastrointestinal Stromal Tumors (GISTs)
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 8, 页码: 3964-3979
作者:
Wang, Qang
;
Liu, Feiyang
;
Wang, Beilei
;
Zou, Fengming
;
Chen, Cheng
;
Liu, Xiaochuan
;
Wang, Aoli
;
Qi, Shuang
;
Wang, Wenchao
;
Qi, Ziping
;
Zhao, Zheng
;
Hu, Zhenquan
;
Wang, Wei
;
Wang, Li
;
Zhang, Shanchun
;
Wang, Yuexiang
;
Liu, Jing
;
Liu, Qingsong
浏览
  |  
Adobe PDF(10221Kb)
  |  
收藏
  |  
浏览/下载:123/72
  |  
提交时间:2017/11/10