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Discovery of N-(5-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)-4-methoxy-2-(4-methyl-1,4-diazepan-1-yl)phenyl)acrylamide (CHMFL-ALK/EGFR-050) as a potent ALK/EGFR dual kinase inhibitor capable of overcoming a variety of ALK/EGFR associated drug resistant mutants in NSCLC 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 139, 期号: 无, 页码: 674-697
作者:  Chen, Yongfei;  Wu, Jiaxin;  Wang, Aoli;  Qi, Ziping;  Jiang, Taoshan;  Chen, Cheng;  Zou, Fengming;  Hu, Chen;  Wang, Wei;  Wu, Hong;  Hu, Zhenquan;  Wang, Wenchao;  Wang, Beilei;  Wang, Li;  Ren, Tao;  Zhang, Shanchun;  Liu, Qingsong;  Liu, Jing
浏览  |  Adobe PDF(12656Kb)  |  收藏  |  浏览/下载:21275/11466  |  提交时间:2018/08/17
Egfr  Alk  Dual Kinase Inhibitor  Non-small Cell Lung Cancer  
JQ1 synergizes with the Bcl-2 inhibitor ABT-263 against MYCN-amplified small cell lung cancer 期刊论文
ONCOTARGET, 2017, 卷号: 8, 期号: 49, 页码: 86312-86324
作者:  Wang, Huogang;  Hong, Bo;  Li, Xuemin;  Deng, Ke;  Li, Hong;  Lui, Vivian Wai Yan;  Lin, Wenchu
浏览  |  Adobe PDF(9738Kb)  |  收藏  |  浏览/下载:92/39  |  提交时间:2018/08/17
Small Cell Lung Cancer  N-myc  Bcl-2  Jq1  Abt-263  
Impacts of lung and tumor volumes on lung dosimetry for nonsmall cell lung cancer 期刊论文
JOURNAL OF APPLIED CLINICAL MEDICAL PHYSICS, 2017, 卷号: 18, 期号: 5, 页码: 22-28
作者:  Lei, Weijie;  Jia, Jing;  Cao, Ruifen;  Song, Jing;  Hu, Liqin
Adobe PDF(297Kb)  |  收藏  |  浏览/下载:88/39  |  提交时间:2019/06/17
lung cancer  intensity-modulated radiotherapy  volumetric-modulated arc therapy  
Kinases Involved in Both Autophagy and Mitosis 期刊论文
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2017, 卷号: 18, 期号: 9, 页码: 1-15
作者:  Li, Zhiyuan;  Zhang, Xin
浏览  |  Adobe PDF(277Kb)  |  收藏  |  浏览/下载:105/48  |  提交时间:2018/08/17
Kinases  Autophagy  Mitosis  Cyclin-dependent Kinases  Aurora  Polo-like Kinases  
A pH-Responsive Yolk-Like Nanoplatform for Tumor Targeted Dual-Mode Magnetic Resonance Imaging and Chemotherapy 期刊论文
ACS NANO, 2017, 卷号: 11, 期号: 7, 页码: 7049-7059
作者:  Sun, Xiao;  Du, Ruohong;  Zhang, Li;  Zhang, Guilong;  Zheng, Xiaojia;  Qian, Junchao;  Tian, Xiaohe;  Zhou, Jiewen;  He, Jiacai;  Wang, Yuanyin;  Wu, Yiqun;  Zhong, Kai;  Cai, Dongqing;  Zou, Duohong;  Wu, Zhengyan
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Yolk-like Fe3o4@gd2o3  Targeted  Dual-mode Mr Imaging Drug Delivery System  Cisplatin  Ph Responsive  Cancer Chemotherapy  
Biocompatible Chitosan-Carbon Dot Hybrid Nanogels for NIR-Imaging-Guided Synergistic Photothermal-Chemo Therapy 期刊论文
ACS APPLIED MATERIALS & INTERFACES, 2017, 卷号: 9, 期号: 22, 页码: 18639-18649
作者:  Wang, Hui;  Mukherjee, Sumit;  Ji, Jinhui;  Banerjee, Probal;  Chen, Qianwang;  Zhou, Shuiqin
浏览  |  Adobe PDF(9178Kb)  |  收藏  |  浏览/下载:96/62  |  提交时间:2018/05/25
Carbon Dots  Chitosan  Cchns  Responsive Release  Nir Imaging  
基于微流控芯片的中性粒细胞运动及趋化性研究 学位论文
, 合肥: 中国科学技术大学, 2017
作者:  杨柯
Adobe PDF(4670Kb)  |  收藏  |  浏览/下载:45/1  |  提交时间:2018/01/18
针对FLT3-ITD阳性急性髓细胞白血病的激酶抑制剂药物学研究 学位论文
, 合肥: 中国科学技术大学, 2017
作者:  王傲莉
Adobe PDF(7111Kb)  |  收藏  |  浏览/下载:138/0  |  提交时间:2018/01/18
EpCAM Inhibition Sensitizes Chemoresistant Leukemia to Immune Surveillance 期刊论文
CANCER RESEARCH, 2017, 卷号: 77, 期号: 2, 页码: 482-493
作者:  Zheng, Xiaohu;  Fan, Xiaolei;  Fu, Binqing;  Zheng, Meijuan;  Zhang, Aimei;  Zhong, Kai;  Yan, Jialai;  Sun, Rui;  Tian, Zhigang;  Wei, Haiming
浏览  |  Adobe PDF(2088Kb)  |  收藏  |  浏览/下载:181/142  |  提交时间:2018/07/04
叶酸受体介导的磁性纳米给药系统的构建及用于肿瘤诊治的实验研究 学位论文
, 合肥: 中国科学技术大学, 2017
作者:  杜若鸿
Adobe PDF(3713Kb)  |  收藏  |  浏览/下载:40/0  |  提交时间:2018/01/18