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中国科学院合肥物质科学研究院机构知识库
Knowledge Management System of Hefei Institute of Physical Science,CAS
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中科院强磁场科学中... [10]
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刘青松 [12]
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Osimertinib successfully combats EGFR-negative glioblastoma cells by inhibiting the MAPK pathway
期刊论文
ACTA PHARMACOLOGICA SINICA, 2020
作者:
Chen, Cheng
;
Cheng, Chuan-dong
;
Wu, Hong
;
Wang, Zuo-wei
;
Wang, Li
;
Jiang, Zong-ru
;
Wang, Ao-li
;
Hu, Chen
;
Dong, Yong-fei
;
Niu, Wan-xiang
;
Qi, Shuang
;
Qi, Zi-ping
;
Liu, Jing
;
Wang, Wen-chao
;
Niu, Chao-shi
;
Liu, Qing-song
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Adobe PDF(3476Kb)
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浏览/下载:91/34
  |  
提交时间:2020/11/26
glioblastoma
osimertinib
temozolamide
MAPK-signaling pathway
MNK
eukaryotic translation initiation factor 4E
Discovery of N-(4-(6-Acetamidopyrimidin-4-yloxy)phenyl)-2-(2-(trifluoromethyl)phenyl)acetamide (CHMFL-FLT3-335) as a Potent FMS-like Tyrosine Kinase 3 Internal Tandem Duplication (FLT3-ITD) Mutant Selective Inhibitor for Acute Myeloid Leukemia
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 2, 页码: 875-892
作者:
Liang, Xiaofei
;
Wang, Beilei
;
Chen, Cheng
;
Wang, Aoli
;
Hu, Chen
;
Zou, Fengming
;
Yu, Kailin
;
Liu, Qingwang
;
Li, Feng
;
Hu, Zhenquan
;
Lu, Tingting
;
Wang, Junjie
;
Wang, Li
;
Weisberg, Ellen L.
;
Li, Lili
;
Xia, Ruixiang
;
Wang, Wenchao
;
Ren, Tao
;
Ge, Jian
;
Liu, Jing
;
Liu, Qinsong
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Adobe PDF(13868Kb)
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浏览/下载:363/319
  |  
提交时间:2020/05/21
Sodium chloride (NaCl) potentiates digoxin-induced anti-tumor activity in small cell lung cancer
期刊论文
CANCER BIOLOGY & THERAPY, 2019, 卷号: 20, 期号: 1, 页码: 52-64
作者:
Deng, Ke
;
Shen, Jiawei
;
Wang, Wei
;
Li, Ming
;
Li, Hong
;
Chen, Cheng
;
Zhao, Huan
;
Zhang, Mei
;
Xue, Tian
;
Liu, Qingsong
;
Lui, Vivian Wai Yan
;
Hong, Bo
;
Lin, Wenchu
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Adobe PDF(3554Kb)
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浏览/下载:66/27
  |  
提交时间:2020/03/31
small cell lung cancer
digoxin
NaCl
cardiac glycosides
ATP1A1
Discovery of 4-((N-(2-(dimethylamino)ethyl)acrylamido)methyl)-N-(4-methyl-3-((4-(pyridin-3-yl)pyrimidin-2-yl)amino)phenyl)benzamide (CHMFL-PDGFR-159) as a highly selective type II PDGFR alpha kinase inhibitor for PDGFR alpha driving chronic eosinophilic leukemia
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 150, 期号: 无, 页码: 366-384
作者:
Wang, Qiang
;
Liu, Feiyang
;
Qi, Shuang
;
Qi, Ziping
;
Yan, Xiao-E.
;
Wang, Beilei
;
Wang, Aoli
;
Wang, Wei
;
Chen, Cheng
;
Liu, Xiaochuan
;
Jiang, Zongru
;
Hu, Zhenquan
;
Wang, Li
;
Wang, Wenchao
;
Ren, Tao
;
Zhang, Shanchun
;
Yun, Cai-Hong
;
Liu, Qingsong
;
Liu, Jing
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  |  
Adobe PDF(5108Kb)
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浏览/下载:588/505
  |  
提交时间:2019/06/10
PDGFR kinase
Type II inhibitor
Kinase inhibitor
CEL
Discovery of 4-((N-(2-(dimethylamino)ethyl)acrylamido)methyl)-N-(4-methyl-3-((4-(pyridin-3-yl)pyrimidin-2-yl)amino)phenyl)benzamide (CHMFL-PDGFR-159) as a highly selective type II PDGFRα kinase inhibi
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018
作者:
Qiang Wang
;
Feiyang Liu
;
Qi S(亓爽)
;
Ziping Qi
;
Beilei Wang
;
Aoli Wang
;
Zongru Jiang
;
Wenchao Wang
;
Qingsong Liu
;
Jing Liu
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  |  
Adobe PDF(5108Kb)
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  |  
浏览/下载:123/51
  |  
提交时间:2020/10/20
Discovery of N-(5-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)-4-methoxy-2-(4-methyl-1,4-diazepan-1-yl)phenyl)acrylamide (CHMFL-ALK/EGFR-050) as a potent ALK/EGFR dual kinase inhibitor capable of overcoming a variety of ALK/EGFR associated drug resistant mutants in NSCLC
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 139, 期号: 无, 页码: 674-697
作者:
Chen, Yongfei
;
Wu, Jiaxin
;
Wang, Aoli
;
Qi, Ziping
;
Jiang, Taoshan
;
Chen, Cheng
;
Zou, Fengming
;
Hu, Chen
;
Wang, Wei
;
Wu, Hong
;
Hu, Zhenquan
;
Wang, Wenchao
;
Wang, Beilei
;
Wang, Li
;
Ren, Tao
;
Zhang, Shanchun
;
Liu, Qingsong
;
Liu, Jing
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  |  
Adobe PDF(12656Kb)
  |  
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  |  
浏览/下载:21274/11466
  |  
提交时间:2018/08/17
Egfr
Alk
Dual Kinase Inhibitor
Non-small Cell Lung Cancer
Simultaneous inhibition of Vps34 kinase would enhance PI3K delta inhibitor cytotoxicity in the B-cell malignancies
期刊论文
ONCOTARGET, 2016, 卷号: 7, 期号: 33, 页码: 53515-53525
作者:
Liu, Xiaochuan
;
Wang, Aoli
;
Liang, Xiaofei
;
Liu, Juanjuan
;
Zou, Fengming
;
Chen, Cheng
;
Zhao, Zheng
;
Deng, Yuanxin
;
Wu, Hong
;
Qi, Ziping
;
Wang, Beilei
;
Wang, Li
;
Liu, Feiyang
;
Xu, Yunhe
;
Wang, Wenchao
;
Fernandes, Stacey M.
;
Stone, Richard M.
;
Galinsky, Ilene A.
;
Brown, Jennifer R.
;
Loh, Teckpeng
;
Griffin, James. D.
;
Zhang, Shanchun
;
Weisberg, Ellen L.
;
Zhang, Xin
;
Liu, Jing
;
Liu, Qingsong
浏览
  |  
Adobe PDF(7625Kb)
  |  
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  |  
浏览/下载:89/37
  |  
提交时间:2017/11/21
Pi3k Delta
Vps34
Combination
Chronic Lymphatic Leukemia
Acute Myeloid Leukemia
Moderate and strong static magnetic fields directly affect EGFR kinase domain orientation to inhibit cancer cell proliferation
期刊论文
ONCOTARGET, 2016, 卷号: 7, 期号: 27, 页码: 41527-41539
作者:
Zhang, Lei
;
Wang, Jihao
;
Wang, HongLei
;
Wang, Wenchao
;
Li, Zhiyuan
;
Liu, Juanjuan
;
Yang, Xingxing
;
Ji, Xinmiao
;
Luo, Yan
;
Hu, Chen
;
Hou, Yubin
;
He, Qianqian
;
Fang, Jun
;
Wang, Junfeng
;
Liu, Qingsong
;
Li, Guohui
;
Lu, Qingyou
;
Zhang, Xin
浏览
  |  
Adobe PDF(11191Kb)
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浏览/下载:93/37
  |  
提交时间:2017/11/21
Egfr
Magnetic Field
Stm
Cancer
Moderate intensity static magnetic fields affect mitotic spindles and increase the antitumor efficacy of 5-FU and Taxol
期刊论文
BIOELECTROCHEMISTRY, 2016, 卷号: 109, 期号: 无, 页码: 31-40
作者:
Luo, Yan
;
Ji, Xinmiao
;
Liu, Juanjuan
;
Li, Zhiyuan
;
Wang, Wenchao
;
Chen, Wei
;
Wang, Junfeng
;
Liu, Qingsong
;
Zhang, Xin
浏览
  |  
Adobe PDF(2812Kb)
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收藏
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浏览/下载:94/48
  |  
提交时间:2017/11/10
Static Magnetic Field
Microtubule
Mitosis
Cancer Cells
5-fluorouracil
Cisplatin
Discovery of N-(34(1-lsonicotinoylpiperidin-4-yl)oxy)-4methylpheny1)-3-(trifluoromethyl)benzamide (CHMFL-KIT-110) as a Selective, Potent, and Orally Available Type II c-KIT Kinase Inhibitor for Gastrointestinal Stromal Tumors (GISTs)
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 8, 页码: 3964-3979
作者:
Wang, Qang
;
Liu, Feiyang
;
Wang, Beilei
;
Zou, Fengming
;
Chen, Cheng
;
Liu, Xiaochuan
;
Wang, Aoli
;
Qi, Shuang
;
Wang, Wenchao
;
Qi, Ziping
;
Zhao, Zheng
;
Hu, Zhenquan
;
Wang, Wei
;
Wang, Li
;
Zhang, Shanchun
;
Wang, Yuexiang
;
Liu, Jing
;
Liu, Qingsong
浏览
  |  
Adobe PDF(10221Kb)
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收藏
  |  
浏览/下载:121/71
  |  
提交时间:2017/11/10