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Discovery of (E)-N-(4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)-3-((3-(2-(pyridin-2-yl)vinyl)-1H-indazol-6-yl)thio)propanamide (CHMFL-ABL-121) as a highly potent ABL kinase inhibitor capable of overcoming a variety of ABL mutants including T315I for chronic myeloid leukemia 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 160, 页码: 61-81
作者:  Liu, Xuesong;  Wang, Beilei;  Chen, Cheng;  Jiang, Zongru;  Hu, Chen;  Wu, Hong;  Zhang, Yicong;  Liu, Xiaochuan;  Wang, Wenliang;  Wang, Junjie;  Hu, Zhenquan;  Wang, Aoli;  Huang, Tao;  Liu, Qingwang;  Wang, Wei;  Wang, Li;  Wang, Wenchao;  Ren, Tao;  Li, Lili;  Xia, Ruixiang;  Ge, Jian;  Liu, Qingsong;  Liu, Jing
Adobe PDF(4593Kb)  |  收藏  |  浏览/下载:190/104  |  提交时间:2019/01/11
ABL kinase  Kinase inhibitor  ABL mutant  CML  
Estimation of carbon impurity from the guard limiter of the lower hybrid wave antenna on EAST tokamak 期刊论文
PLASMA PHYSICS AND CONTROLLED FUSION, 2018, 卷号: 60, 期号: 12, 页码: 11
作者:  Ou, Jing;  Xiang, Nong;  Liu, Liang;  Men, Zongzheng;  Zhang, Ling;  Mao, Songtao;  Chen, Meiwen
Adobe PDF(1532Kb)  |  收藏  |  浏览/下载:111/55  |  提交时间:2019/01/11
physical sputtering  chemical erosion  hot spot  plasma sheath  
Strategy Design and Transient Analysis of ITER PPEN Transformer On-Load Tap Changer During Converter Operation 期刊论文
JOURNAL OF FUSION ENERGY, 2018, 卷号: 37, 期号: 6, 页码: 346-353
作者:  Fan, Renjing;  Fu, Peng;  Tao, Jun;  Gao, Ge;  Song, Zhiquan;  Huang, Liansheng;  Chen, Xiaojiao;  Li, Jinchao
收藏  |  浏览/下载:32/0  |  提交时间:2019/12/25
ITER  Coil power supply  OLTC control  Hysteresis band  Converter operation robustness  
Observation of tungsten impurities induced 2/1 snake fluctuations and their interactions with discrete double BAE pairs on EAST 期刊论文
NUCLEAR FUSION, 2018, 卷号: 58, 期号: 12, 页码: 8
作者:  Xu, Ming;  Zhou, T.;  Xu, L. Q.;  Hu, L. Q.;  Duan, Y. M.;  Liu, Y.;  Zhang, L.;  Shi, T. H.;  Li, Y. Y.;  Lyu, B.;  Zhao, H. L.;  Chen, Y. J.;  Zhang, Y.;  Huang, J.;  Xu, G. S.;  Sun, Y. W.;  Zhang, X. D.;  Wan, B. N.
收藏  |  浏览/下载:38/0  |  提交时间:2019/12/25
2/1 snake fluctuations  discrete double BAEs  discrete spectra  tearing modes  
Sequential deposition route to efficient Sb2S3 solar cells 期刊论文
JOURNAL OF MATERIALS CHEMISTRY A, 2018, 卷号: 6, 期号: 43, 页码: 21320-21326
作者:  Zhang, Lijian;  Wu, Chunyan;  Liu, Weifeng;  Yang, Shangfeng;  Wang, Mingtai;  Chen, Tao;  Zhu, Changfei
Adobe PDF(1174Kb)  |  收藏  |  浏览/下载:133/78  |  提交时间:2019/01/11
Full-inorganic Sb-2(S, Se)(3) solar cells using carbon as both hole selection material and electrode 期刊论文
ELECTROCHIMICA ACTA, 2018, 卷号: 290, 页码: 457-464
作者:  Wang, Weihuang;  Chen, Guilin;  Wang, Zhezhe;  Wang, Ke;  Chen, Shuiyuan;  Huang, Zhigao;  Wang, Xiaomin;  Chen, Tao;  Zhu, Changfei;  Kong, Xiangkai
收藏  |  浏览/下载:33/0  |  提交时间:2019/12/25
Sb-2(S,Se)(3)  Full-inorganic  Selenization  Solar cell  Carbon  
Experimental study on the magnetic coherent mode in the H-mode pedestal of EAST 期刊论文
NUCLEAR FUSION, 2018, 卷号: 58, 期号: 11, 页码: 20
作者:  Chen, Ran;  Zhang, Heng;  Xu, Guosheng;  Zhou, Chu;  Li, Yongliang;  Ye, Yang;  Shi, Tonghui;  Liu, Haiqing;  Zhang, Tao;  Gao, Wei;  Liu, Yong;  Lyu, Bo;  Zang, Qing;  Xu, Jichan;  Feng, Wei;  Liu, Adi;  Wang, Liang;  Qian, Jinping;  Ding, Siye;  Wang, Huiqian;  Wu, Xingquan;  Yang, Qingquan;  Hu, Guanghai;  Liang, Yunfeng;  Gong, Xianzu;  Wan, Baonian
收藏  |  浏览/下载:59/0  |  提交时间:2019/12/20
magnetic coherent mode  pedestal  edge-localized mode  divertor particle flux  
Discovery of 4-(((4-(5-chloro-2-(((1s,4s)-4-((2-methoxyethyl)amino) cyclohexyl)amino)pyridin-4-yl)thiazol-2-yl)amino)methyl) tetrahydro-2H-pyran-4-carbonitrile (JSH-150) as a novel highly selective and potent CDK9 kinase inhibitor 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 158, 页码: 896-916
作者:  Wang, Beilei;  Wu, Jiaxin;  Wu, Yun;  Chen, Cheng;  Zou, Fengming;  Wang, Aoli;  Wu, Hong;  Hu, Zhenquan;  Jiang, Zongru;  Liu, Qingwang;  Wang, Wei;  Zhang, Yicong;  Liu, Feiyang;  Zhao, Ming;  Hu, Jie;  Huang, Tao;  Ge, Juan;  Wang, Li;  Ren, Tao;  Wang, Yuxin;  Liu, Jing;  Liu, Qingsong
收藏  |  浏览/下载:25/0  |  提交时间:2019/12/25
CDK9  Kinase inhibitor  Structure-activity relationship  Leukemia  
Disruption of Chromosomal Architecture of cox2 Locus Sensitizes Lung Cancer Cells to Radiotherapy 期刊论文
MOLECULAR THERAPY, 2018, 卷号: 26, 期号: 10, 页码: 2456-2465
作者:  Sun, Yuxiang;  Dai, Hui;  Chen, Shaopeng;  Zhang, Yajun;  Wu, Tao;  Cao, Xianbin;  Zhao, Guoping;  Xu, An;  Wang, Jun;  Wu, Lijun
收藏  |  浏览/下载:25/0  |  提交时间:2019/12/25
Observation of toroidal Alfven eigenmode excited by energetic electrons induced by static magnetic perturbations in the EAST tokamak 期刊论文
NUCLEAR FUSION, 2018, 卷号: 58, 期号: 10, 页码: 5
作者:  Chu, N.;  Sun, Y.;  Gu, S.;  Wang, H. H.;  Hu, Y. J.;  Shi, T. H.;  Chen, D. L.;  Gu, X.;  He, K. Y.;  Jia, M.;  Lin, S. Y.;  Liu, H. Q.;  Qian, J. P.;  Ren, J.;  Shen, B.;  Ti, A.;  Wang, S. X.;  Xie, J. L.;  Xu, M.;  Xue, M. M.;  Yan, N.;  Zang, Q.;  Zeng, L.;  Zhang, J. Z.;  Zhang, T.;  Zhang, Y.;  Zhong, G. Q.;  Zhou, C.;  Zhou, R. J.
收藏  |  浏览/下载:48/0  |  提交时间:2019/11/11
magnetic perturbation  toroidal Alfven eignenmode  reconnection  magnetic island  energetic electron