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Discovery and characterization of a novel highly potent and selective type II native and drug-resistant V299L mutant BCR-ABL inhibitor (CHMFL-ABL-039) for Chronic Myeloid Leukemia (CML) 期刊论文
CANCER BIOLOGY & THERAPY, 2019, 卷号: 20, 期号: 6, 页码: 877-885
作者:  Wu, Jiaxin;  Wang, Aoli;  Li, Xixiang;  Chen, Cheng;  Qi, Ziping;  Hu, Chen;  Wang, Wenliang;  Wu, Hong;  Huang, Tao;  Zhao, Ming;  Wang, Wenchao;  Hu, Zhenquan;  Liu, Qingwang;  Wang, Beilei;  Wang, Li;  Li, Lili;  Ge, Jian;  Ren, Tao;  Xia, Ruixiang;  Liu, Jing
收藏  |  浏览/下载:52/0  |  提交时间:2019/11/27
BCR-ABL  PDGFR  chronic myeloid leukemia  kinase inhibitor  
Giant antiferromagnetic negative thermal expansion in (MnNiGe)(1-x)(MnCoSn)(x) compounds 期刊论文
JOURNAL OF ALLOYS AND COMPOUNDS, 2019, 卷号: 782, 期号: 无, 页码: 881-886
作者:  Zhu, Feng;  Lin, Jianchao;  Zhang, Xuekai;  Li, Longfu;  Yang, Cheng;  Wang, Meng;  Wu, Ying;  Tong, Peng;  Song, Wenhai;  Sun, Yuping
浏览  |  Adobe PDF(2150Kb)  |  收藏  |  浏览/下载:89/40  |  提交时间:2020/05/21
Negative thermal expansion  Martensitic transformation  AFM ground state  Magnetostriction  Thermal conductivity  
Discovery of N-(4-(6-Acetamidopyrimidin-4-yloxy)phenyl)-2-(2-(trifluoromethyl)phenyl)acetamide (CHMFL-FLT3-335) as a Potent FMS-like Tyrosine Kinase 3 Internal Tandem Duplication (FLT3-ITD) Mutant Selective Inhibitor for Acute Myeloid Leukemia 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 2, 页码: 875-892
作者:  Liang, Xiaofei;  Wang, Beilei;  Chen, Cheng;  Wang, Aoli;  Hu, Chen;  Zou, Fengming;  Yu, Kailin;  Liu, Qingwang;  Li, Feng;  Hu, Zhenquan;  Lu, Tingting;  Wang, Junjie;  Wang, Li;  Weisberg, Ellen L.;  Li, Lili;  Xia, Ruixiang;  Wang, Wenchao;  Ren, Tao;  Ge, Jian;  Liu, Jing;  Liu, Qinsong
浏览  |  Adobe PDF(13868Kb)  |  收藏  |  浏览/下载:369/319  |  提交时间:2020/05/21
Synthesis, physical properties, and annealing investigation of new layered Bi-chalcogenide LaOBiHgS3 期刊论文
CHINESE PHYSICS B, 2019, 卷号: 28, 期号: 1, 页码: 4
作者:  Yu, Yi;  Wang, Chunchang;  Li, Liang;  Li, Qiuju;  Cheng, Chao;  Wang, Shuting;  Zhang, Changjin
浏览  |  Adobe PDF(392Kb)  |  收藏  |  浏览/下载:79/46  |  提交时间:2020/03/31
thermoelectric material  Bi-chalcogenide  post annealing  
Molecular-scale investigation of fluoride sorption mechanism by nanosized hydroxyapatite using F-19 solid-state NMR spectroscopy 期刊论文
JOURNAL OF COLLOID AND INTERFACE SCIENCE, 2019
作者:  Ren, Chao;  Yu, Zhiwu;  Phillips, Brian L.;  Wang, Hongtao;  Ji, Junfeng;  Pan, Bingcai;  Li, Wei
浏览  |  Adobe PDF(3062Kb)  |  收藏  |  浏览/下载:80/41  |  提交时间:2020/10/29
Enhancement of thermoelectric properties by fluorine doping in LaO1-xFxBiPbS3 期刊论文
CERAMICS INTERNATIONAL, 2019, 卷号: 45, 期号: 1, 页码: 817-821
作者:  Yu, Yi;  Wang, Chunchang;  Li, Qiuju;  Cheng, Chao;  Wang, Shuting;  Zhang, Changjin
收藏  |  浏览/下载:36/0  |  提交时间:2019/12/25
Thermoelectric properties  Low-dimensional material  BiS2-basedmaterial  Power factor  Phase separation  
Repurposing cabozantinib to GISTs: Overcoming multiple imatinib-resistant cKIT mutations including gatekeeper and activation loop mutants in GISTs preclinical models 期刊论文
CANCER LETTERS, 2019, 页码: 105-114
作者:  Lu, Tingting;  Chen, Cheng;  Wang, Aoli;  Jiang, Zongru;  Qi, Ziping;  Hu, Zhenquan;  Hu, Chen;  Liu, Feiyang;  Wang, Wenliang;  Wu, Hong;  Wang, Beilei;  Wang, Li;  Qi, Shuang;  Wu, Jiaxin;  Wang, Wenchao;  Tang, Jun;  Yan, Hezhong;  Bai, Mingfeng;  Liu, Qingsong;  Liu, Jing
收藏  |  浏览/下载:23/0  |  提交时间:2020/07/14
cKIT T670I mutant  Activation loop mutants  Drug resistance  
NIR-responsive carbon-based nanocarriers for switchable on/off drug release and synergistic cancer therapy 期刊论文
JOURNAL OF MATERIALS CHEMISTRY B, 2018, 卷号: 6, 期号: 47, 页码: 7794-7799
作者:  Nie, Rongrong;  Liu, Hongji;  Hu, Lin;  Gu, Xinyu;  Qian, Junchao;  Wang, Hui
收藏  |  浏览/下载:25/0  |  提交时间:2019/12/25
Magnetic field-induced electronic phase transition in the Dirac semimetal state of black phosphorus under pressure 期刊论文
SCIENCE BULLETIN, 2018, 卷号: 63, 期号: 23, 页码: 1539-1544
作者:  Sun, Zeliang;  Xiang, Ziji;  Wang, Zhongyi;  Zhang, Jinglei;  Ma, Long;  Wang, Naizhou;  Shang, Chao;  Meng, Fanbao;  Zou, Liangjian;  Zhang, Yuanbo;  Chen, Xianhui
收藏  |  浏览/下载:32/0  |  提交时间:2019/12/25
Black phosphorus  High magnetic field  Quantum limit  Electron phase transition  
Discovery of (E)-N-(4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)-3-((3-(2-(pyridin-2-yl)vinyl)-1H-indazol-6-yl)thio)propanamide (CHMFL-ABL-121) as a highly potent ABL kinase inhibitor capable of overcoming a variety of ABL mutants including T315I for chronic myeloid leukemia 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 160, 页码: 61-81
作者:  Liu, Xuesong;  Wang, Beilei;  Chen, Cheng;  Jiang, Zongru;  Hu, Chen;  Wu, Hong;  Zhang, Yicong;  Liu, Xiaochuan;  Wang, Wenliang;  Wang, Junjie;  Hu, Zhenquan;  Wang, Aoli;  Huang, Tao;  Liu, Qingwang;  Wang, Wei;  Wang, Li;  Wang, Wenchao;  Ren, Tao;  Li, Lili;  Xia, Ruixiang;  Ge, Jian;  Liu, Qingsong;  Liu, Jing
Adobe PDF(4593Kb)  |  收藏  |  浏览/下载:190/104  |  提交时间:2019/01/11
ABL kinase  Kinase inhibitor  ABL mutant  CML