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中国科学院合肥物质科学研究院机构知识库
Knowledge Management System of Hefei Institute of Physical Science,CAS
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中科院强磁场科学中心 [9]
作者
刘青松 [10]
吴宏 [10]
王文超 [10]
王傲莉 [9]
齐紫平 [7]
刘小川 [6]
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CHMFL-26 is a highly potent irreversible HER2 inhibitor for use in the treatment of HER2-positive and HER2-mutant cancers
期刊论文
ACTA PHARMACOLOGICA SINICA, 2022
作者:
Cao, Jiang-yan
;
Qi, Shuang
;
Wu, Hong
;
Wang, Ao-li
;
Liu, Qing-wang
;
Li, Xi-xiang
;
Wang, Bei-lei
;
Ge, Juan
;
Zou, Feng-ming
;
Chen, Cheng
;
Wang, Jun-jie
;
Hu, Chen
;
Liu, Jing
;
Wang, Wen-chao
;
Liu, Qing-song
收藏
  |  
浏览/下载:92/0
  |  
提交时间:2022/03/28
HER2
breast cancers
gastric cancers
irreversible inhibitor
drug resistance
Discovery of 1-(4-(4-Amino-3-(4-(2-morpholinoethoxy)-phenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)phenyl)-3-(5-(tert-butyl)isoxazol-3-yl)urea (CHMFL-FLT3-213) as a Highly Potent Type II FLT3 Kinase Inhibitor Capable of Overcoming a Variety of FLT3 Kinase Mutants in FLT3-ITD Positive AML
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 20, 页码: 8407-8424
作者:
Wang, Aoli
;
Li, Xixiang
;
Chen, Cheng
;
Wu, Hong
;
Qi, Ziping
;
Hu, Chen
;
Yu, Kailin
;
Wu, Jiaxin
;
Liu, Juan
;
Liu, Xiaochuan
;
Hu, Zhenquan
;
Wang, Wei
;
Wang, Wenliang
;
Wang, Wenchao
;
Wang, Li
;
Wang, Beilei
;
Liu, Qingwang
;
Li, Lili
;
Ge, Jian
;
Ren, Tao
;
Zhang, Shanchun
;
Xia, Ruixiang
;
Liu, Jing
;
Liu, Qingsong
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  |  
Adobe PDF(10028Kb)
  |  
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  |  
浏览/下载:78/31
  |  
提交时间:2019/06/17
Discovery of 2-((3-Acrylamido-4-methylphenyl)amino)-N-(2-methyl5-(3,4,5-trimethoxybenzamido)phenyI)-4-(methylamino)pyrimidine-5-carboxamide (CHMFL-BMX-078) as a Highly Potent and Selective Type II Irreversible Bone Marrow Kinase in the X Chromosome (BMX) Kinase Inhibitor
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 5, 页码: 1793-1816
作者:
Liang, Xiaofei
;
Lv, Fengchao
;
Wang, Beilei
;
Yu, Kailin
;
Wu, Hong
;
Qi, Ziping
;
Jiang, Zongru
;
Chen, Cheng
;
Wang, Aoli
;
Miao, Weili
;
Wang, Wenchao
;
Hu, Zhenquan
;
Liu, Juan
;
Liu, Xiaochuan
;
Zhao, Zheng
;
Wang, Li
;
Zhang, Shanchuan
;
Ye, Zi
;
Wang, Chu
;
Ren, Tao
;
Wang, Yinsheng
;
Liu, Qingsong
;
Liu, Jing
浏览
  |  
Adobe PDF(5919Kb)
  |  
收藏
  |  
浏览/下载:17292/7523
  |  
提交时间:2018/07/04
Discovery and characterization of a novel irreversible EGFR mutants selective and potent kinase inhibitor CHMFL-EGFR-26 with a distinct binding mode
期刊论文
ONCOTARGET, 2017, 卷号: 8, 期号: 11, 页码: 18359-18372
作者:
Hu, Chen
;
Wang, Aoli
;
Wu, Hong
;
Qi, Ziping
;
Li, Xixiang
;
Yan, Xiao-E
;
Chen, Cheng
;
Yu, Kailin
;
Zou, Fengming
;
Wang, Wenchao
;
Wang, Wei
;
Wu, Jiaxin
;
Liu, Juan
;
Wang, Beilei
;
Wang, Li
;
Ren, Tao
;
Zhang, Shanchun
;
Yun, Cai-Hong
;
Liu, Jing
;
Liu, Qingsong
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  |  
Adobe PDF(6153Kb)
  |  
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  |  
浏览/下载:176/45
  |  
提交时间:2018/07/04
Egfr
Egfrt790m
Nsclc
Kinase Inhibitors
Drug Resistance
Discovery of N-((1-(4-(3-(3-((6,7-Dimethoxyquinolin-3-yl)oxy)phenyl)ureido)-2-(trifluoromethyl)phenyl)piperidin-4-yl)methyl)propionamide (CHMFL-KIT-8140) as a Highly Potent Type II Inhibitor Capable of Inhibiting the T670I "Gatekeeper" Mutant of cKIT Kinase
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 18, 页码: 8456-8472
作者:
Li, Binhua
;
Wang, Aoli
;
Liu, Juan
;
Qi, Ziping
;
Liu, Xiaochuan
;
Yu, Kailin
;
Wu, Hong
;
Chen, Cheng
;
Hu, Chen
;
Wang, Wenchao
;
Wu, Jiaxin
;
Hu, Zhenquan
;
Ye, Ling
;
Zou, Fengming
;
Liu, Feiyang
;
Wang, Beilei
;
Wang, Li
;
Ren, Tao
;
Zhang, Shaojuan
;
Bai, Mingfeng
;
Zhang, Shanchun
;
Liu, Jing
;
Liu, Qingsong
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  |  
Adobe PDF(2856Kb)
  |  
收藏
  |  
浏览/下载:1400/1298
  |  
提交时间:2017/11/21
Simultaneous inhibition of Vps34 kinase would enhance PI3K delta inhibitor cytotoxicity in the B-cell malignancies
期刊论文
ONCOTARGET, 2016, 卷号: 7, 期号: 33, 页码: 53515-53525
作者:
Liu, Xiaochuan
;
Wang, Aoli
;
Liang, Xiaofei
;
Liu, Juanjuan
;
Zou, Fengming
;
Chen, Cheng
;
Zhao, Zheng
;
Deng, Yuanxin
;
Wu, Hong
;
Qi, Ziping
;
Wang, Beilei
;
Wang, Li
;
Liu, Feiyang
;
Xu, Yunhe
;
Wang, Wenchao
;
Fernandes, Stacey M.
;
Stone, Richard M.
;
Galinsky, Ilene A.
;
Brown, Jennifer R.
;
Loh, Teckpeng
;
Griffin, James. D.
;
Zhang, Shanchun
;
Weisberg, Ellen L.
;
Zhang, Xin
;
Liu, Jing
;
Liu, Qingsong
浏览
  |  
Adobe PDF(7625Kb)
  |  
收藏
  |  
浏览/下载:93/37
  |  
提交时间:2017/11/21
Pi3k Delta
Vps34
Combination
Chronic Lymphatic Leukemia
Acute Myeloid Leukemia
Characterization of selective and potent PI3K delta inhibitor (PI3KD-IN-015) for B-Cell malignances
期刊论文
ONCOTARGET, 2016, 卷号: 7, 期号: 22, 页码: 32641-32651
作者:
Liu, Xiaochuan
;
Wang, Aoli
;
Liang, Xiaofei
;
Chen, Cheng
;
Liu, Juanjuan
;
Zhao, Zheng
;
Wu, Hong
;
Deng, Yuanxin
;
Wang, Li
;
Wang, Beilei
;
Wu, Jiaxin
;
Liu, Feiyang
;
Fernandes, Stacey M.
;
Adamia, Sophia
;
Stone, Richard M.
;
Galinsky, Ilene A.
;
Brown, Jennifer R.
;
Griffin, James D.
;
Zhang, Shanchun
;
Loh, Teckpeng
;
Zhang, Xin
;
Wang, Wenchao
;
Weisberg, Ellen L.
;
Liu, Jing
;
Liu, Qingsong
浏览
  |  
Adobe PDF(5138Kb)
  |  
收藏
  |  
浏览/下载:79/28
  |  
提交时间:2017/11/16
Pi3k Delta
Leukemia
B-cell Malignances
Pi3k
Kinase Inhibitors
Dual Inhibition of AKT/FLT3-ITD by A674563 Overcomes FLT3 Ligand-Induced Drug Resistance in FLT3-ITD positive AML
期刊论文
ONCOTARGET, 2016, 卷号: 7, 期号: 20, 页码: 29131-29142
作者:
Wang, Aoli
;
Wu, Hong
;
Chen, Cheng
;
Hu, Chen
;
Qi, Ziping
;
Wang, Wenchao
;
Yu, Kailin
;
Liu, Xiaochuan
;
Zou, Fengming
;
Zhao, Zheng
;
Wu, Jiaxin
;
Liu, Juan
;
Liu, Feiyang
;
Wang, Li
;
Stone, Richard M.
;
Galinksy, Ilene A.
;
Griffin, James D.
;
Zhang, Shanchun
;
Weisberg, Ellen L.
;
Liu, Jing
;
Liu, Qingsong
浏览
  |  
Adobe PDF(4786Kb)
  |  
收藏
  |  
浏览/下载:132/35
  |  
提交时间:2017/11/16
Acute Myeloid Leukemia
Flt3-itd
Akt
A6745763
Flt3-ligand
Ammonia Induces Autophagy through Dopamine Receptor D3 and MTOR
期刊论文
PLOS ONE, 2016, 卷号: 11, 期号: 4, 页码: 1-24
作者:
Li, Zhiyuan
;
Ji, Xinmiao
;
Wang, Wenchao
;
Liu, Juanjuan
;
Liang, Xiaofei
;
Wu, Hong
;
Liu, Jing
;
Eggert, Ulrike S.
;
Liu, Qingsong
;
Zhang, Xin
浏览
  |  
Adobe PDF(7380Kb)
  |  
收藏
  |  
浏览/下载:91/43
  |  
提交时间:2017/11/10
Discovery of (R)-1-(3-(4-Amino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)-2-(dimethylamino)ethanone (CHMFL-FLT3-122) as a Potent and Orally Available FLT3 Kinase Inhibitor for FLT3-ITD Positive Acute Myeloid Leukemia
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2015, 卷号: 58, 期号: 24, 页码: 9625-9638
作者:
Li, Xixiang
;
Wang, Aoli
;
Yu, Kailin
;
Qi, Ziping
;
Chen, Cheng
;
Wang, Wenchao
;
Hu, Chen
;
Wu, Hong
;
Wu, Jiaxin
;
Zhao, Zheng
;
Liu, Juan
;
Zou, Fengming
;
Wang, Li
;
Wang, Beilei
;
Wang, Wei
;
Zhang, Shanchun
;
Liu, Jing
;
Liu, Qingsong
浏览
  |  
Adobe PDF(6123Kb)
  |  
收藏
  |  
浏览/下载:158/100
  |  
提交时间:2017/10/25