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中国科学院合肥物质科学研究院机构知识库
Knowledge Management System of Hefei Institute of Physical Science,CAS
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刘青松 [8]
王文超 [8]
王傲莉 [8]
胡晨 [7]
齐紫平 [5]
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(本次检索基于用户作品认领结果)
浏览/检索结果:
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Inhibition of the deubiquitinating enzyme USP47 as a novel targeted therapy for hematologic malignancies expressing mutant EZH2
期刊论文
LEUKEMIA, 2022
作者:
Yang, Jing
;
Weisberg, Ellen L.
;
Qi, Shuang
;
Ni, Wei
;
Mei, Husheng
;
Wang, Zuowei
;
Meng, Chengcheng
;
Zhang, Shengzhe
;
Hou, Mingqi
;
Qi, Ziping
;
Wang, Aoli
;
Jiang, Yunyun
;
Jiang, Zongru
;
Huang, Tao
;
Liu, Qingwang
;
Magin, Robert S.
;
Doherty, Laura
;
Wang, Wenchao
;
Liu, Jing
;
Buhrlage, Sara J.
;
Liu, Qingsong
;
Griffin, James D.
收藏
  |  
浏览/下载:76/0
  |  
提交时间:2022/02/14
Discovery of a highly potent kinase inhibitor capable of overcoming multiple imatinib-resistant ABL mutants for chronic myeloid leukemia (CML)
期刊论文
EUROPEAN JOURNAL OF PHARMACOLOGY, 2021, 卷号: 897
作者:
Lu, Tingting
;
Cao, Jiangyan
;
Zou, Fengming
;
Li, Xixiang
;
Wang, Aoli
;
Wang, Wenliang
;
Liang, Huamin
;
Liu, Qingwang
;
Hu, Chen
;
Chen, Cheng
;
Hu, Zhenquan
;
Wang, Wenchao
;
Li, Lili
;
Ge, Jian
;
Shen, Yang
;
Ren, Tao
;
Liu, Jing
;
Xia, Ruixiang
;
Liu, Qingsong
收藏
  |  
浏览/下载:69/0
  |  
提交时间:2021/04/26
BCR-ABL
ABL mutants
Chronic myeloid leukemia
Kinase inhibitor
Imatinib resistance
Selectively targeting FLT3-ITD mutants over FLT3-wt by a novel inhibitor for acute myeloid leukemia
期刊论文
HAEMATOLOGICA, 2021, 卷号: 106
作者:
Wang, Aoli
;
Hu, Chen
;
Chen, Cheng
;
Liang, Xiaofei
;
Wang, Beilei
;
Zou, Fengming
;
Yu, Kailin
;
Li, Feng
;
Liu, Qingwang
;
Qi, Ziping
;
Wang, Junjie
;
Wang, Wenliang
;
Wang, Li
;
Weisberg, Ellen L.
;
Wang, Wenchao
;
Li, Lili
;
Ge, Jian
;
Xia, Ruixiang
;
Liu, Jing
;
Liu, Qingsong
收藏
  |  
浏览/下载:50/0
  |  
提交时间:2021/04/26
Discovery of a highly selective VEGFR2 kinase inhibitor CHMFL-VEGFR2-002 as a novel anti-angiogenesis agent
期刊论文
ACTA PHARMACEUTICA SINICA B, 2020, 卷号: 10
作者:
Jiang, Zongru
;
Wang, Li
;
Liu, Xuesong
;
Chen, Cheng
;
Wang, Beilei
;
Wang, Wenliang
;
Hu, Chen
;
Yu, Kailin
;
Qi, Ziping
;
Liu, Qingwang
;
Wang, Aoli
;
Liu, Jing
;
Hong, Guangchen
;
Wang, Wenchao
;
Liu, Qingsong
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2020/11/26
Cancer
VEGFR2 kinase
Kinase inhibitor
Angiogenesis
Inhibitor selectivity
Discovery and characterization of a novel highly potent and selective type II native and drug-resistant V299L mutant BCR-ABL inhibitor (CHMFL-ABL-039) for Chronic Myeloid Leukemia (CML)
期刊论文
CANCER BIOLOGY & THERAPY, 2019, 卷号: 20, 期号: 6, 页码: 877-885
作者:
Wu, Jiaxin
;
Wang, Aoli
;
Li, Xixiang
;
Chen, Cheng
;
Qi, Ziping
;
Hu, Chen
;
Wang, Wenliang
;
Wu, Hong
;
Huang, Tao
;
Zhao, Ming
;
Wang, Wenchao
;
Hu, Zhenquan
;
Liu, Qingwang
;
Wang, Beilei
;
Wang, Li
;
Li, Lili
;
Ge, Jian
;
Ren, Tao
;
Xia, Ruixiang
;
Liu, Jing
收藏
  |  
浏览/下载:52/0
  |  
提交时间:2019/11/27
BCR-ABL
PDGFR
chronic myeloid leukemia
kinase inhibitor
Discovery of N-(4-(6-Acetamidopyrimidin-4-yloxy)phenyl)-2-(2-(trifluoromethyl)phenyl)acetamide (CHMFL-FLT3-335) as a Potent FMS-like Tyrosine Kinase 3 Internal Tandem Duplication (FLT3-ITD) Mutant Selective Inhibitor for Acute Myeloid Leukemia
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 2, 页码: 875-892
作者:
Liang, Xiaofei
;
Wang, Beilei
;
Chen, Cheng
;
Wang, Aoli
;
Hu, Chen
;
Zou, Fengming
;
Yu, Kailin
;
Liu, Qingwang
;
Li, Feng
;
Hu, Zhenquan
;
Lu, Tingting
;
Wang, Junjie
;
Wang, Li
;
Weisberg, Ellen L.
;
Li, Lili
;
Xia, Ruixiang
;
Wang, Wenchao
;
Ren, Tao
;
Ge, Jian
;
Liu, Jing
;
Liu, Qinsong
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  |  
Adobe PDF(13868Kb)
  |  
收藏
  |  
浏览/下载:369/319
  |  
提交时间:2020/05/21
Discovery of (E)-N-(4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)-3-((3-(2-(pyridin-2-yl)vinyl)-1H-indazol-6-yl)thio)propanamide (CHMFL-ABL-121) as a highly potent ABL kinase inhibitor capable of overcoming a variety of ABL mutants including T315I for chronic myeloid leukemia
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 160, 页码: 61-81
作者:
Liu, Xuesong
;
Wang, Beilei
;
Chen, Cheng
;
Jiang, Zongru
;
Hu, Chen
;
Wu, Hong
;
Zhang, Yicong
;
Liu, Xiaochuan
;
Wang, Wenliang
;
Wang, Junjie
;
Hu, Zhenquan
;
Wang, Aoli
;
Huang, Tao
;
Liu, Qingwang
;
Wang, Wei
;
Wang, Li
;
Wang, Wenchao
;
Ren, Tao
;
Li, Lili
;
Xia, Ruixiang
;
Ge, Jian
;
Liu, Qingsong
;
Liu, Jing
Adobe PDF(4593Kb)
  |  
收藏
  |  
浏览/下载:190/104
  |  
提交时间:2019/01/11
ABL kinase
Kinase inhibitor
ABL mutant
CML
Discovery of 1-(4-(4-Amino-3-(4-(2-morpholinoethoxy)-phenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)phenyl)-3-(5-(tert-butyl)isoxazol-3-yl)urea (CHMFL-FLT3-213) as a Highly Potent Type II FLT3 Kinase Inhibitor Capable of Overcoming a Variety of FLT3 Kinase Mutants in FLT3-ITD Positive AML
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 20, 页码: 8407-8424
作者:
Wang, Aoli
;
Li, Xixiang
;
Chen, Cheng
;
Wu, Hong
;
Qi, Ziping
;
Hu, Chen
;
Yu, Kailin
;
Wu, Jiaxin
;
Liu, Juan
;
Liu, Xiaochuan
;
Hu, Zhenquan
;
Wang, Wei
;
Wang, Wenliang
;
Wang, Wenchao
;
Wang, Li
;
Wang, Beilei
;
Liu, Qingwang
;
Li, Lili
;
Ge, Jian
;
Ren, Tao
;
Zhang, Shanchun
;
Xia, Ruixiang
;
Liu, Jing
;
Liu, Qingsong
浏览
  |  
Adobe PDF(10028Kb)
  |  
收藏
  |  
浏览/下载:78/31
  |  
提交时间:2019/06/17