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中国科学院合肥物质科学研究院机构知识库
Knowledge Management System of Hefei Institute of Physical Science,CAS
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中科院强磁场科学中... [10]
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王薇 [10]
刘青松 [10]
吴宏 [10]
王文超 [10]
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Structure-activity relationship investigation for benzonaphthyridinone derivatives as novel potent Bruton's tyrosine kinase (BTK) irreversible inhibitors
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 137, 页码: 545-557
作者:
Wang, Beilei
;
Deng, Yuanxin
;
Chen, Yongfei
;
Yu, Kailin
;
Wang, Aoli
;
Liang, Qianmao
;
Wang, Wei
;
Chen, Cheng
;
Wu, Hong
;
Hu, Chen
;
Miao, Weili
;
Hur, Wooyoung
;
Wang, Wenchao
;
Hu, Zhenquan
;
Weisberg, Ellen L.
;
Wang, Jinhua
;
Ren, Tao
;
Wang, Yinsheng
;
Gray, Nathanael S.
;
Liu, Qingsong
;
Liu, Jing
收藏
  |  
浏览/下载:347/0
  |  
提交时间:2018/08/16
Btk
Kinase Inhibitor
Irreversible Inhibitor
Structure-activity Relationship
B-cell Lymphoma
Discovery of (R)-1-(3-(4-Amino-3-(3-chloro-4-(pyridin-2-ylmethoxy)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-one (CHMFL-EGFR-202) as a Novel Irreversible EGFR Mutant Kinase Inhibitor with a Distinct Binding Mode
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 7, 页码: 2944-2962
作者:
Wang, Aoli
;
Li, Xixiang
;
Wu, Hong
;
Zou, Fengming
;
Yan, Xiao-E
;
Chen, Cheng
;
Hu, Chen
;
Yu, Kailin
;
Wang, Wenchao
;
Zhao, Peng
;
Wu, Jiaxin
;
Qi, Ziping
;
Wang, Wei
;
Wang, Beilei
;
Wang, Li
;
Ren, Tao
;
Zhang, Shanchun
;
Yun, Cai-Hong
;
Liu, Jing
;
Liu, Qingsong
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2018/07/26
Discovery of (R)-1-(3-(4-Amino-3-(3-chloro-4-(pyridin-2-ylmethoxy)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-one (CHMFL-EGFR-202) as a Novel Irreversible EGFR Mutant Kinase Inhibitor with a Distinct Binding Mode
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 7, 页码: 2944-2962
作者:
Wang, Aoli
;
Li, Xixiang
;
Wu, Hong
;
Zou, Fengming
;
Yan, Xiao-E
;
Chen, Cheng
;
Hu, Chen
;
Yu, Kailin
;
Wang, Wenchao
;
Zhao, Peng
;
Wu, Jiaxin
;
Qi, Ziping
;
Wang, Wei
;
Wang, Beilei
;
Wang, Li
;
Ren, Tao
;
Zhang, Shanchun
;
Yun, Cai-Hong
;
Liu, Jing
;
Liu, Qingsong
收藏
  |  
浏览/下载:48/0
  |  
提交时间:2018/07/26
Discovery of (R)-1-(3-(4-Amino-3-(3-chloro-4-(pyridin-2-ylmethoxy)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-one (CHMFL-EGFR-202) as a Novel Irreversible EGFR Mutant Kinase Inhibitor with a Distinct Binding Mode
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 7, 页码: 2944-2962
作者:
Wang, Aoli
;
Li, Xixiang
;
Wu, Hong
;
Zou, Fengming
;
Yan, Xiao-E
;
Chen, Cheng
;
Hu, Chen
;
Yu, Kailin
;
Wang, Wenchao
;
Zhao, Peng
;
Wu, Jiaxin
;
Qi, Ziping
;
Wang, Wei
;
Wang, Beilei
;
Wang, Li
;
Ren, Tao
;
Zhang, Shanchun
;
Yun, Cai-Hong
;
Liu, Jing
;
Liu, Qingsong
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2018/07/26
Discovery of (R)-1-(3-(4-Amino-3-(3-chloro-4-(pyridin-2-ylmethoxy)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-one (CHMFL-EGFR-202) as a Novel Irreversible EGFR Mutant Kinase Inhibitor with a Distinct Binding Mode
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 7, 页码: 2944-2962
作者:
Wang, Aoli
;
Li, Xixiang
;
Wu, Hong
;
Zou, Fengming
;
Yan, Xiao-E
;
Chen, Cheng
;
Hu, Chen
;
Yu, Kailin
;
Wang, Wenchao
;
Zhao, Peng
;
Wu, Jiaxin
;
Qi, Ziping
;
Wang, Wei
;
Wang, Beilei
;
Wang, Li
;
Ren, Tao
;
Zhang, Shanchun
;
Yun, Cai-Hong
;
Liu, Jing
;
Liu, Qingsong
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2018/07/26
Discovery of (R)-1-(3-(4-Amino-3-(3-chloro-4-(pyridin-2-ylmethoxy)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-one (CHMFL-EGFR-202) as a Novel Irreversible EGFR Mutant Kinase Inhibitor with a Distinct Binding Mode
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 7, 页码: 2944-2962
作者:
Wang, Aoli
;
Li, Xixiang
;
Wu, Hong
;
Zou, Fengming
;
Yan, Xiao-E
;
Chen, Cheng
;
Hu, Chen
;
Yu, Kailin
;
Wang, Wenchao
;
Zhao, Peng
;
Wu, Jiaxin
;
Qi, Ziping
;
Wang, Wei
;
Wang, Beilei
;
Wang, Li
;
Ren, Tao
;
Zhang, Shanchun
;
Yun, Cai-Hong
;
Liu, Jing
;
Liu, Qingsong
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2018/07/26
Discovery of (R)-1-(3-(4-Amino-3-(3-chloro-4-(pyridin-2-ylmethoxy)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-one (CHMFL-EGFR-202) as a Novel Irreversible EGFR Mutant Kinase Inhibitor with a Distinct Binding Mode
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 7, 页码: 2944-2962
作者:
Wang, Aoli
;
Li, Xixiang
;
Wu, Hong
;
Zou, Fengming
;
Yan, Xiao-E
;
Chen, Cheng
;
Hu, Chen
;
Yu, Kailin
;
Wang, Wenchao
;
Zhao, Peng
;
Wu, Jiaxin
;
Qi, Ziping
;
Wang, Wei
;
Wang, Beilei
;
Wang, Li
;
Ren, Tao
;
Zhang, Shanchun
;
Yun, Cai-Hong
;
Liu, Jing
;
Liu, Qingsong
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2018/07/26
Discovery of (R)-1-(3-(4-Amino-3-(3-chloro-4-(pyridin-2-ylmethoxy)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-one (CHMFL-EGFR-202) as a Novel Irreversible EGFR Mutant Kinase Inhibitor with a Distinct Binding Mode
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 7, 页码: 2944-2962
作者:
Wang, Aoli
;
Li, Xixiang
;
Wu, Hong
;
Zou, Fengming
;
Yan, Xiao-E
;
Chen, Cheng
;
Hu, Chen
;
Yu, Kailin
;
Wang, Wenchao
;
Zhao, Peng
;
Wu, Jiaxin
;
Qi, Ziping
;
Wang, Wei
;
Wang, Beilei
;
Wang, Li
;
Ren, Tao
;
Zhang, Shanchun
;
Yun, Cai-Hong
;
Liu, Jing
;
Liu, Qingsong
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2018/07/26
Discovery of (R)-1-(3-(4-Amino-3-(3-chloro-4-(pyridin-2-ylmethoxy)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-one (CHMFL-EGFR-202) as a Novel Irreversible EGFR Mutant Kinase Inhibitor with a Distinct Binding Mode
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 7, 页码: 2944-2962
作者:
Wang, Aoli
;
Li, Xixiang
;
Wu, Hong
;
Zou, Fengming
;
Yan, Xiao-E
;
Chen, Cheng
;
Hu, Chen
;
Yu, Kailin
;
Wang, Wenchao
;
Zhao, Peng
;
Wu, Jiaxin
;
Qi, Ziping
;
Wang, Wei
;
Wang, Beilei
;
Wang, Li
;
Ren, Tao
;
Zhang, Shanchun
;
Yun, Cai-Hong
;
Liu, Jing
;
Liu, Qingsong
收藏
  |  
浏览/下载:47/0
  |  
提交时间:2018/07/26
Discovery and characterization of a novel irreversible EGFR mutants selective and potent kinase inhibitor CHMFL-EGFR-26 with a distinct binding mode
期刊论文
ONCOTARGET, 2017, 卷号: 8, 期号: 11, 页码: 18359-18372
作者:
Hu, Chen
;
Wang, Aoli
;
Wu, Hong
;
Qi, Ziping
;
Li, Xixiang
;
Yan, Xiao-E
;
Chen, Cheng
;
Yu, Kailin
;
Zou, Fengming
;
Wang, Wenchao
;
Wang, Wei
;
Wu, Jiaxin
;
Liu, Juan
;
Wang, Beilei
;
Wang, Li
;
Ren, Tao
;
Zhang, Shanchun
;
Yun, Cai-Hong
;
Liu, Jing
;
Liu, Qingsong
浏览
  |  
Adobe PDF(6153Kb)
  |  
收藏
  |  
浏览/下载:178/46
  |  
提交时间:2018/07/04
Egfr
Egfrt790m
Nsclc
Kinase Inhibitors
Drug Resistance