×
验证码:
换一张
忘记密码?
记住我
切换中国科技网通行证登录
×
切换中国科技网通行证登录
登录
中文版
|
English
中国科学院合肥物质科学研究院机构知识库
Knowledge Management System of Hefei Institute of Physical Science,CAS
登录
注册
ALL
ORCID
题名
作者
学科领域
关键词
文献类型
出处
收录类别
出版者
发表日期
存缴日期
资助项目
学科门类
学习讨论厅
图片搜索
粘贴图片网址
首页
研究单元&专题
作者
文献类型
学科分类
知识图谱
新闻&公告
在结果中检索
研究单元&专题
中科院强磁场科学中... [15]
中科院安徽光学精密机... [7]
医学 [2]
作者
刘飞扬 [18]
刘青松 [16]
王文超 [14]
王傲莉 [12]
齐紫平 [9]
亓爽 [8]
更多...
发表日期
2022 [1]
2020 [1]
2019 [2]
2018 [3]
2017 [2]
2016 [7]
更多...
语种
英语 [14]
出处
JOURNAL OF... [4]
ONCOTARGET [4]
EUROPEAN J... [3]
JOURNAL OF... [2]
JOURNAL OF... [2]
ACS CHEMIC... [1]
更多...
资助项目
National N... [3]
Natural Sc... [3]
China Post... [2]
China Post... [2]
Frontier S... [2]
National N... [2]
更多...
资助机构
China "Tho... [6]
Chinese Ac... [5]
"Hundred T... [3]
Anhui Prov... [3]
CAS/SAFEA ... [3]
China Post... [3]
更多...
收录类别
SCI [15]
摘要
文献类型
期刊论文 [25]
学位论文 [1]
×
知识图谱
HFCAS OpenIR
开始提交
已提交作品
待认领作品
已认领作品
未提交全文
收藏管理
QQ客服
官方微博
反馈留言
浏览/检索结果:
共26条,第1-10条
帮助
只显示已认领条目
已选(
0
)
清除
条数/页:
5
10
15
20
25
30
35
40
45
50
55
60
65
70
75
80
85
90
95
100
排序方式:
请选择
发表日期升序
发表日期降序
WOS被引频次升序
WOS被引频次降序
提交时间升序
提交时间降序
期刊影响因子升序
期刊影响因子降序
题名升序
题名降序
作者升序
作者降序
A novel patient-derived organoid model for triple-negative breast cancer patients with residual disease after neoadjuvant chemotherapy for screening personalized drugs.
期刊论文
JOURNAL OF CLINICAL ONCOLOGY, 2022, 卷号: 40
作者:
Liu, Feiyang
;
Ma, Dandan
;
Liu, Qingsong
;
Qi, Xiaowei
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2022/12/23
Network-based analysis with primary cells reveals drug response landscape of acute myeloid leukemia
期刊论文
EXPERIMENTAL CELL RESEARCH, 2020, 卷号: 393
作者:
Chen, Cheng
;
Wang, Li
;
Li, Lili
;
Wang, Aoli
;
Huang, Tao
;
Hu, Jie
;
Zhao, Ming
;
Liu, Feiyang
;
Qi, Shuang
;
Hu, Chen
;
Wang, Wenliang
;
Liu, Jing
;
Ge, Jian
;
Xia, Ruixiang
;
Wang, Wenchao
;
Liu, Qingsong
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2020/11/26
Acute myeloid leukemia (AML)
Drug response
Gene mutations
Discovery of 2-(4-Chloro-3-(trifluoromethyl)phenyl)-N-(4-((6,7-dimethoxyquinolin-4-yl)oxy)phenyl)acetamide (CHMFL-KIT-64) as a Novel Orally Available Potent Inhibitor against Broad-Spectrum Mutants of
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019
作者:
Yun Wu
;
Beilei Wang
;
Junjie Wang
;
Qi S(亓爽)
;
Fengming Zou
;
Ziping Qi
;
Feiyang Liu
;
Wenchao Wang
;
Qingsong Liu
;
Jing Liu
浏览
  |  
Adobe PDF(5207Kb)
  |  
收藏
  |  
浏览/下载:123/63
  |  
提交时间:2020/10/20
Repurposing cabozantinib to GISTs: Overcoming multiple imatinib-resistant cKIT mutations including gatekeeper and activation loop mutants in GISTs preclinical models
期刊论文
CANCER LETTERS, 2019, 页码: 105-114
作者:
Lu, Tingting
;
Chen, Cheng
;
Wang, Aoli
;
Jiang, Zongru
;
Qi, Ziping
;
Hu, Zhenquan
;
Hu, Chen
;
Liu, Feiyang
;
Wang, Wenliang
;
Wu, Hong
;
Wang, Beilei
;
Wang, Li
;
Qi, Shuang
;
Wu, Jiaxin
;
Wang, Wenchao
;
Tang, Jun
;
Yan, Hezhong
;
Bai, Mingfeng
;
Liu, Qingsong
;
Liu, Jing
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2020/07/14
cKIT T670I mutant
Activation loop mutants
Drug resistance
Discovery of 4-(((4-(5-chloro-2-(((1s,4s)-4-((2-methoxyethyl)amino) cyclohexyl)amino)pyridin-4-yl)thiazol-2-yl)amino)methyl) tetrahydro-2H-pyran-4-carbonitrile (JSH-150) as a novel highly selective and potent CDK9 kinase inhibitor
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 158, 页码: 896-916
作者:
Wang, Beilei
;
Wu, Jiaxin
;
Wu, Yun
;
Chen, Cheng
;
Zou, Fengming
;
Wang, Aoli
;
Wu, Hong
;
Hu, Zhenquan
;
Jiang, Zongru
;
Liu, Qingwang
;
Wang, Wei
;
Zhang, Yicong
;
Liu, Feiyang
;
Zhao, Ming
;
Hu, Jie
;
Huang, Tao
;
Ge, Juan
;
Wang, Li
;
Ren, Tao
;
Wang, Yuxin
;
Liu, Jing
;
Liu, Qingsong
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2019/12/25
CDK9
Kinase inhibitor
Structure-activity relationship
Leukemia
Discovery of 4-((N-(2-(dimethylamino)ethyl)acrylamido)methyl)-N-(4-methyl-3-((4-(pyridin-3-yl)pyrimidin-2-yl)amino)phenyl)benzamide (CHMFL-PDGFR-159) as a highly selective type II PDGFR alpha kinase inhibitor for PDGFR alpha driving chronic eosinophilic leukemia
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 150, 期号: 无, 页码: 366-384
作者:
Wang, Qiang
;
Liu, Feiyang
;
Qi, Shuang
;
Qi, Ziping
;
Yan, Xiao-E.
;
Wang, Beilei
;
Wang, Aoli
;
Wang, Wei
;
Chen, Cheng
;
Liu, Xiaochuan
;
Jiang, Zongru
;
Hu, Zhenquan
;
Wang, Li
;
Wang, Wenchao
;
Ren, Tao
;
Zhang, Shanchun
;
Yun, Cai-Hong
;
Liu, Qingsong
;
Liu, Jing
浏览
  |  
Adobe PDF(5108Kb)
  |  
收藏
  |  
浏览/下载:588/505
  |  
提交时间:2019/06/10
PDGFR kinase
Type II inhibitor
Kinase inhibitor
CEL
Discovery of 4-((N-(2-(dimethylamino)ethyl)acrylamido)methyl)-N-(4-methyl-3-((4-(pyridin-3-yl)pyrimidin-2-yl)amino)phenyl)benzamide (CHMFL-PDGFR-159) as a highly selective type II PDGFRα kinase inhibi
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018
作者:
Qiang Wang
;
Feiyang Liu
;
Qi S(亓爽)
;
Ziping Qi
;
Beilei Wang
;
Aoli Wang
;
Zongru Jiang
;
Wenchao Wang
;
Qingsong Liu
;
Jing Liu
浏览
  |  
Adobe PDF(5108Kb)
  |  
收藏
  |  
浏览/下载:123/51
  |  
提交时间:2020/10/20
Gemcitabine and Chk1 Inhibitor AZD7762 Synergistically Suppress the Growth of Lkb1-Deficient Lung Adenocarcinoma
期刊论文
CANCER RESEARCH, 2017, 卷号: 77, 期号: 18, 页码: 5068-5076
作者:
Liu, Yan
;
Li, Yuyang
;
Wang, Xiaoen
;
Liu, Feiyang
;
Gao, Peng
;
Quinn, Max M.
;
Li, Fei
;
Merlino, Ashley A.
;
Benes, Cyril
;
Liu, Qingsong
;
Gray, Nathanael S.
;
Wong, Kwok-Kin
收藏
  |  
浏览/下载:47/0
  |  
提交时间:2018/08/16
Discovery of 4-Methyl-N-(44(4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)-3-((1-nicotinoylpiperidin-4-y1)oxy)benzamide (CHMFL-ABL/KIT-155) as a Novel Highly Potent Type II ABL/KIT Dual Kinase Inhibitor with a Distinct Hinge Binding
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 1, 页码: 273-289
作者:
Wang, Qiang
;
Liu, Feiyang
;
Wang, Beilei
;
Zou, Fengming
;
Qi, Ziping
;
Chen, Cheng
;
Yu, Kailin
;
Hu, Chen
;
Qi, Shuang
;
Wang, Wenchao
;
Hu, Zhenquan
;
Liu, Juan
;
Wang, Wei
;
Wang, Li
;
Liang, Qianmao
;
Zhang, Shanchun
;
Ren, Tao
;
Liu, Qingsong
;
Liu, Jing
浏览
  |  
Adobe PDF(3516Kb)
  |  
收藏
  |  
浏览/下载:99/57
  |  
提交时间:2018/07/04
Discovery of N-((1-(4-(3-(3-((6,7-Dimethoxyquinolin-3-yl)oxy)phenyl)ureido)-2-(trifluoromethyl)phenyl)piperidin-4-yl)methyl)propionamide (CHMFL-KIT-8140) as a Highly Potent Type II Inhibitor Capable of Inhibiting the T670I "Gatekeeper" Mutant of cKIT Kinase
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 18, 页码: 8456-8472
作者:
Li, Binhua
;
Wang, Aoli
;
Liu, Juan
;
Qi, Ziping
;
Liu, Xiaochuan
;
Yu, Kailin
;
Wu, Hong
;
Chen, Cheng
;
Hu, Chen
;
Wang, Wenchao
;
Wu, Jiaxin
;
Hu, Zhenquan
;
Ye, Ling
;
Zou, Fengming
;
Liu, Feiyang
;
Wang, Beilei
;
Wang, Li
;
Ren, Tao
;
Zhang, Shaojuan
;
Bai, Mingfeng
;
Zhang, Shanchun
;
Liu, Jing
;
Liu, Qingsong
浏览
  |  
Adobe PDF(2856Kb)
  |  
收藏
  |  
浏览/下载:1395/1298
  |  
提交时间:2017/11/21