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中国科学院合肥物质科学研究院机构知识库
Knowledge Management System of Hefei Institute of Physical Science,CAS
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CHMFL-26 is a highly potent irreversible HER2 inhibitor for use in the treatment of HER2-positive and HER2-mutant cancers
期刊论文
ACTA PHARMACOLOGICA SINICA, 2022
Authors:
Cao, Jiang-yan
;
Qi, Shuang
;
Wu, Hong
;
Wang, Ao-li
;
Liu, Qing-wang
;
Li, Xi-xiang
;
Wang, Bei-lei
;
Ge, Juan
;
Zou, Feng-ming
;
Chen, Cheng
;
Wang, Jun-jie
;
Hu, Chen
;
Liu, Jing
;
Wang, Wen-chao
;
Liu, Qing-song
Favorite
  |  
View/Download:24/0
  |  
Submit date:2022/03/28
HER2
breast cancers
gastric cancers
irreversible inhibitor
drug resistance
Inhibition of the deubiquitinating enzyme USP47 as a novel targeted therapy for hematologic malignancies expressing mutant EZH2
期刊论文
LEUKEMIA, 2022
Authors:
Yang, Jing
;
Weisberg, Ellen L.
;
Qi, Shuang
;
Ni, Wei
;
Mei, Husheng
;
Wang, Zuowei
;
Meng, Chengcheng
;
Zhang, Shengzhe
;
Hou, Mingqi
;
Qi, Ziping
;
Wang, Aoli
;
Jiang, Yunyun
;
Jiang, Zongru
;
Huang, Tao
;
Liu, Qingwang
;
Magin, Robert S.
;
Doherty, Laura
;
Wang, Wenchao
;
Liu, Jing
;
Buhrlage, Sara J.
;
Liu, Qingsong
;
Griffin, James D.
Favorite
  |  
View/Download:25/0
  |  
Submit date:2022/02/14
An overview of kinase downregulators and recent advances in discovery approaches
期刊论文
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2021, 卷号: 6
Authors:
Wang, Beilei
;
Wu, Hong
;
Hu, Chen
;
Wang, Haizhen
;
Liu, Jing
;
Wang, Wenchao
;
Liu, Qingsong
Favorite
  |  
View/Download:16/0
  |  
Submit date:2022/01/25
Iodine cation bridged graphene sheets with strengthened interface combination for electromagnetic wave absorption
期刊论文
CARBON, 2021, 卷号: 183
Authors:
Li, Qingsong
;
Li, Shitong
;
Liu, Qiangchun
;
Liu, Xiaofang
;
Shui, Jianglan
;
Kong, Xiangkai
Favorite
  |  
View/Download:6/0
  |  
Submit date:2021/11/15
Iodine cation
Microwave absorbing
Graphene
Targeting chaperon protein HSP70 as a novel therapeutic strategy for FLT3-ITD-positive acute myeloid leukemia
期刊论文
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2021, 卷号: 6
Authors:
Hu, Chen
;
Zou, Fengming
;
Wang, Aoli
;
Miao, Weili
;
Liang, Qianmao
;
Weisberg, Ellen L.
;
Wang, Yinsheng
;
Liu, Jing
;
Wang, Wenchao
;
Liu, Qingsong
Favorite
  |  
View/Download:5/0
  |  
Submit date:2021/11/01
Nanocrystal-loaded liposome for targeted delivery of poorly water-soluble antitumor drugs with high drug loading and stability towards efficient cancer therapy
期刊论文
INTERNATIONAL JOURNAL OF PHARMACEUTICS, 2021, 卷号: 599
Authors:
Liang, Huamin
;
Zou, Fengming
;
Liu, Qingwang
;
Wang, Beilei
;
Fu, Liyi
;
Liang, Xiaofei
;
Liu, Jing
;
Liu, Qingsong
Favorite
  |  
View/Download:6/0
  |  
Submit date:2021/05/17
Liposome
Drug nanocrystal
Core-shell
Drug delivery
Tumor therapy
BCR-ABL
Discovery of a highly potent kinase inhibitor capable of overcoming multiple imatinib-resistant ABL mutants for chronic myeloid leukemia (CML)
期刊论文
EUROPEAN JOURNAL OF PHARMACOLOGY, 2021, 卷号: 897
Authors:
Lu, Tingting
;
Cao, Jiangyan
;
Zou, Fengming
;
Li, Xixiang
;
Wang, Aoli
;
Wang, Wenliang
;
Liang, Huamin
;
Liu, Qingwang
;
Hu, Chen
;
Chen, Cheng
;
Hu, Zhenquan
;
Wang, Wenchao
;
Li, Lili
;
Ge, Jian
;
Shen, Yang
;
Ren, Tao
;
Liu, Jing
;
Xia, Ruixiang
;
Liu, Qingsong
Favorite
  |  
View/Download:11/0
  |  
Submit date:2021/04/26
BCR-ABL
ABL mutants
Chronic myeloid leukemia
Kinase inhibitor
Imatinib resistance
Selectively targeting FLT3-ITD mutants over FLT3-wt by a novel inhibitor for acute myeloid leukemia
期刊论文
HAEMATOLOGICA, 2021, 卷号: 106
Authors:
Wang, Aoli
;
Hu, Chen
;
Chen, Cheng
;
Liang, Xiaofei
;
Wang, Beilei
;
Zou, Fengming
;
Yu, Kailin
;
Li, Feng
;
Liu, Qingwang
;
Qi, Ziping
;
Wang, Junjie
;
Wang, Wenliang
;
Wang, Li
;
Weisberg, Ellen L.
;
Wang, Wenchao
;
Li, Lili
;
Ge, Jian
;
Xia, Ruixiang
;
Liu, Jing
;
Liu, Qingsong
Favorite
  |  
View/Download:8/0
  |  
Submit date:2021/04/26
Dynamic folding modulation generates FGF21 variant against diabetes
期刊论文
EMBO REPORTS, 2021, 卷号: 22
Authors:
Zhu, Lei
;
Zhao, Hongxin
;
Liu, Juanjuan
;
Cai, Hao
;
Wu, Bo
;
Liu, Zhijun
;
Zhou, Shu
;
Liu, Qingsong
;
Li, Xiaokun
;
Bao, Bin
;
Liu, Jian
;
Dai, Han
;
Wang, Junfeng
Favorite
  |  
View/Download:3/0
  |  
Submit date:2021/08/30
anti‐
diabetes
disulfide bond mutation
FGF21
folding dynamics
NMR
Activating microwave absorption performance by reduced graphene oxide-borophene heterostructure
期刊论文
COMPOSITES PART A-APPLIED SCIENCE AND MANUFACTURING, 2020, 卷号: 138
Authors:
Wang, Shipeng
;
Li, Qingsong
;
Hu, Kang
;
Liu, Qiangchun
;
Liu, Xiaofang
;
Kong, Xiangkai
Favorite
  |  
View/Download:5/0
  |  
Submit date:2020/11/30
Graphene
Borophene
Metal-free
Microwave absorption