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中国科学院合肥物质科学研究院机构知识库
Knowledge Management System of Hefei Institute of Physical Science,CAS
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Inhibition of the deubiquitinating enzyme USP47 as a novel targeted therapy for hematologic malignancies expressing mutant EZH2
期刊论文
LEUKEMIA, 2022
Authors:
Yang, Jing
;
Weisberg, Ellen L.
;
Qi, Shuang
;
Ni, Wei
;
Mei, Husheng
;
Wang, Zuowei
;
Meng, Chengcheng
;
Zhang, Shengzhe
;
Hou, Mingqi
;
Qi, Ziping
;
Wang, Aoli
;
Jiang, Yunyun
;
Jiang, Zongru
;
Huang, Tao
;
Liu, Qingwang
;
Magin, Robert S.
;
Doherty, Laura
;
Wang, Wenchao
;
Liu, Jing
;
Buhrlage, Sara J.
;
Liu, Qingsong
;
Griffin, James D.
Favorite
  |  
View/Download:25/0
  |  
Submit date:2022/02/14
Nanocrystal-loaded liposome for targeted delivery of poorly water-soluble antitumor drugs with high drug loading and stability towards efficient cancer therapy
期刊论文
INTERNATIONAL JOURNAL OF PHARMACEUTICS, 2021, 卷号: 599
Authors:
Liang, Huamin
;
Zou, Fengming
;
Liu, Qingwang
;
Wang, Beilei
;
Fu, Liyi
;
Liang, Xiaofei
;
Liu, Jing
;
Liu, Qingsong
Favorite
  |  
View/Download:6/0
  |  
Submit date:2021/05/17
Liposome
Drug nanocrystal
Core-shell
Drug delivery
Tumor therapy
BCR-ABL
Discovery of a highly potent kinase inhibitor capable of overcoming multiple imatinib-resistant ABL mutants for chronic myeloid leukemia (CML)
期刊论文
EUROPEAN JOURNAL OF PHARMACOLOGY, 2021, 卷号: 897
Authors:
Lu, Tingting
;
Cao, Jiangyan
;
Zou, Fengming
;
Li, Xixiang
;
Wang, Aoli
;
Wang, Wenliang
;
Liang, Huamin
;
Liu, Qingwang
;
Hu, Chen
;
Chen, Cheng
;
Hu, Zhenquan
;
Wang, Wenchao
;
Li, Lili
;
Ge, Jian
;
Shen, Yang
;
Ren, Tao
;
Liu, Jing
;
Xia, Ruixiang
;
Liu, Qingsong
Favorite
  |  
View/Download:11/0
  |  
Submit date:2021/04/26
BCR-ABL
ABL mutants
Chronic myeloid leukemia
Kinase inhibitor
Imatinib resistance
Synthesis, biological evaluation and structure-activity relationship of novel dichloroacetophenones targeting pyruvate dehydrogenase kinases with potent anticancer activity
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 214
Authors:
Xu, Biao
;
Wang, Zhi-Peng
;
Liu, Qingwang
;
Yang, Xiaohong
;
Li, Xuemin
;
Huang, Ding
;
Qiu, Yanfei
;
Tam, Kin Yip
;
Zhang, Shao-Lin
;
He, Yun
Favorite
  |  
View/Download:18/0
  |  
Submit date:2021/04/26
Pyruvate dehydrogenase kinase
Proliferation
Cancer metabolism
Structure-activity relationship
Selectively targeting FLT3-ITD mutants over FLT3-wt by a novel inhibitor for acute myeloid leukemia
期刊论文
HAEMATOLOGICA, 2021, 卷号: 106
Authors:
Wang, Aoli
;
Hu, Chen
;
Chen, Cheng
;
Liang, Xiaofei
;
Wang, Beilei
;
Zou, Fengming
;
Yu, Kailin
;
Li, Feng
;
Liu, Qingwang
;
Qi, Ziping
;
Wang, Junjie
;
Wang, Wenliang
;
Wang, Li
;
Weisberg, Ellen L.
;
Wang, Wenchao
;
Li, Lili
;
Ge, Jian
;
Xia, Ruixiang
;
Liu, Jing
;
Liu, Qingsong
Favorite
  |  
View/Download:9/0
  |  
Submit date:2021/04/26
An ultra-long circulating nanoparticle for reviving a highly selective BCR-ABL inhibitor in long-term effective and safe treatment of chronic myeloid leukemia
期刊论文
NANOMEDICINE-NANOTECHNOLOGY BIOLOGY AND MEDICINE, 2020, 卷号: 29
Authors:
Fu, Liyi
;
Zou, Fengming
;
Liu, Qingwang
;
Wang, Beilei
;
Wang, Junqing
;
Liang, Huamin
;
Liang, Xiaofei
;
Liu, Jing
;
Shi, Jinjun
;
Liu, Qingsong
Favorite
  |  
View/Download:1/0
  |  
Submit date:2020/11/30
Chronic myeloid leukemia
BCR-ABL
Long-circulating nanoparticle
Drug delivery
Discovery of a highly potent and selective Bruton's tyrosine kinase inhibitor avoiding impairment of ADCC effects for B-cell non-Hodgkin lymphoma
期刊论文
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2020, 卷号: 5
Authors:
Liu, Juan
;
Liang, Qianmao
;
Wang, Aoli
;
Zou, Fengming
;
Qi, Ziping
;
Yu, Kailin
;
Liu, Qingwang
;
Chen, Cheng
;
Liu, Jing
;
Liu, Qingsong
Favorite
  |  
View/Download:9/0
  |  
Submit date:2020/11/30
Repurposing of Kinase Inhibitors for Treatment of COVID-19
期刊论文
PHARMACEUTICAL RESEARCH, 2020, 卷号: 37
Authors:
Weisberg, Ellen
;
Parent, Alexander
;
Yang, Priscilla L.
;
Sattler, Martin
;
Liu, Qingsong
;
Liu, Qingwang
;
Wang, Jinhua
;
Meng, Chengcheng
;
Buhrlage, Sara J.
;
Gray, Nathanael
;
Griffin, James D.
Favorite
  |  
View/Download:12/0
  |  
Submit date:2020/10/26
Coronavirus
SARS-CoV-2
SARS-CoV
MERS-CoV
kinase inhibitors
pharmacokinetics
antiviral therapy
COVID-19
Discovery of a highly selective VEGFR2 kinase inhibitor CHMFL-VEGFR2-002 as a novel anti-angiogenesis agent
期刊论文
ACTA PHARMACEUTICA SINICA B, 2020, 卷号: 10
Authors:
Jiang, Zongru
;
Wang, Li
;
Liu, Xuesong
;
Chen, Cheng
;
Wang, Beilei
;
Wang, Wenliang
;
Hu, Chen
;
Yu, Kailin
;
Qi, Ziping
;
Liu, Qingwang
;
Wang, Aoli
;
Liu, Jing
;
Hong, Guangchen
;
Wang, Wenchao
;
Liu, Qingsong
Favorite
  |  
View/Download:9/0
  |  
Submit date:2020/11/26
Cancer
VEGFR2 kinase
Kinase inhibitor
Angiogenesis
Inhibitor selectivity
Discovery of 6 '-chloro-N-methyl-5 '-(phenylsulfonamido)-[3,3 '-bipyridine]-5-carboxamide (CHMFL-PI4K-127) as a novel Plasmodium falciparum PI(4)K inhibitor with potent antimalarial activity against both blood and liver stages of Plasmodium
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 188
Authors:
Liang, Xiaofei
;
Jiang, Zongru
;
Huang, Zhenghui
;
Li, Feng
;
Chen, Cheng
;
Hu, Chen
;
Wang, Wenliang
;
Hu, Zhenquan
;
Liu, Qingwang
;
Wang, Beilei
;
Wang, Li
;
Qi, Ziping
;
Liu, Jing
;
Jiang, Lubin
;
Liu, Qingsong
Favorite
  |  
View/Download:6/0
  |  
Submit date:2020/11/26
PI4K kinase
Kinase inhibitor
Malaria
Blood stage
Liver stage